Water

Water

SCHEMBL12002467

O.O=P(O)(O)Oc1cccc2ccccc12.[NaH]

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3A known ✓ Q14432 1/20 0.49
PTGS1 known ✓ P23219 1/20 0.45
MEN1 known ✓ O00255 1/20 0.44
INPPL1 O15357 3/20 0.55
INPP5A Q14642 3/20 0.55
INPP5B P32019 2/20 0.55
SRC P12931 3/20 0.49
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 3/20 0.49
HSD17B10 Q99714 3/20 0.49
HPGD P15428 2/20 0.49
USP2 O75604 1/20 0.49
HTT P42858 1/20 0.48
TDP1 Q9NUW8 1/20 0.46
OGG1 O15527 1/20 0.45
PGR P06401 1/20 0.45
GAA P10253 1/20 0.45
MAPK1 P28482 1/20 0.45
ACP3 P15309 1/20 0.44
BTN3A1 O00481 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL29202854 0.98 INPPL1 (0.57) INPPL1INPP5AINPP5BSRCALDH1A1
SCHEMBL28237202 0.98 INPPL1 (0.57) INPPL1INPP5AINPP5BSRCALDH1A1
SCHEMBL2544707 0.98 INPPL1 (0.57) INPPL1INPP5AINPP5BSRCALDH1A1
SCHEMBL29618036 0.96 INPPL1 (0.59) INPPL1INPP5AINPP5BSRCALDH1A1
SCHEMBL60472 0.96 INPPL1 (0.59) INPPL1INPP5AINPP5BSRCALDH1A1
Potassium SCHEMBL30820065 0.94 INPPL1 (0.57) INPPL1INPP5AINPP5BSRCALDH1A1
SCHEMBL11322823 0.94 INPPL1 (0.57) INPPL1INPP5AINPP5BSRCALDH1A1
Alcohol SCHEMBL28262288 0.89 INPPL1 (0.52) INPPL1INPP5AINPP5BSRCALDH1A1
Biphenyl SCHEMBL28810841 0.89 INPPL1 (0.52) INPPL1INPP5AINPP5BSRCALDH1A1
Guanidine SCHEMBL28303470 0.89 INPPL1 (0.52) INPPL1INPP5AINPP5BSRCALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12576474-B2 Modification method of polyurethane, polyurethane, polishing pad, and modification method of polishing pad KURARAY CO., LTD. (JP) 2026-03-17 US disclosed
US-20240342858-A1 MODIFICATION METHOD OF POLYURETHANE, POLYURETHANE, POLISHING PAD, AND MODIFICATION METHOD OF POLISHING PAD KURARAY CO., LTD. (JP) 2024-10-17 US disclosed
US-12109665-B2 Modification method of polyurethane, polyurethane, polishing pad, and modification method of polishing pad KURARAY CO., LTD. (JP) 2024-10-08 US disclosed
CN-112105667-B Method for modifying polyurethane, polishing pad and method for modifying polishing pad 株式会社可乐丽 2023-01-10 CN disclosed
US-20210276143-A1 MODIFICATION METHOD OF POLYURETHANE, POLYURETHANE, POLISHING PAD, AND MODIFICATION METHOD OF POLISHING PAD KURARAY CO., LTD. (JP) 2021-09-09 US disclosed
CN-112930383-A Composition, film, laminated structure, light-emitting device, and display 住友化学株式会社 2021-06-08 CN disclosed
CN-112912464-A Composition, film, laminated structure, light-emitting device, and display 住友化学株式会社 2021-06-04 CN disclosed
CN-112912462-A Particle, composition, film, laminated structure, light-emitting device, and display 住友化学株式会社 2021-06-04 CN disclosed
CN-112912444-A Composition, film, laminated structure, light-emitting device, and display 住友化学株式会社 2021-06-04 CN disclosed
CN-112888763-A Particle, composition, film, laminated structure, light-emitting device, and display 住友化学株式会社 2021-06-01 CN disclosed
CN-111655818-A Composition, film, laminate structure, light-emitting device, and display 住友化学株式会社 2020-09-11 CN disclosed
WO-2020085513-A1 PARTICLE, COMPOSITION, FILM, LAMINATED STRUCTURE, LIGHT-EMITTING DEVICE, AND DISPLAY 住友化学株式会社 2020-04-30 WO disclosed
WO-2020085361-A1 PARTICLES, COMPOSITION, FILM, LAYERED STRUCTURE, LIGHT-EMITTING DEVICE, AND DISPLAY 住友化学株式会社 2020-04-30 WO disclosed
WO-2020085363-A1 COMPOSITION, FILM, LAMINATE STRUCTURE, LIGHT-EMITTING DEVICE, AND DISPLAY 住友化学株式会社 2020-04-30 WO disclosed
WO-2020085516-A1 COMPOSITION, FILM, LAMINATED STRUCTURE, LIGHT-EMITTING DEVICE, AND DISPLAY 住友化学株式会社 2020-04-30 WO disclosed
WO-2020085514-A1 COMPOSITION, FILM, LAMINATE STRUCTURE, LIGHT-EMITTING DEVICE, AND DISPLAY 住友化学株式会社 2020-04-30 WO disclosed
EP-2678040-A1 A SYSTEM FOR CARGO DELIVERY INTO THE CELLS Cepep III AB (SE) 2014-01-01 EP disclosed
WO-2012145398-A1 DIAGNOSTIC TEST FOR SCHISTOSOMA HAEMATOBIUM EASTERN VIRGINIA MEDICAL SCHOOL (US) 2012-10-26 WO disclosed
WO-2012113846-A1 A SYSTEM FOR CARGO DELIVERY INTO THE CELLS CEPEP III AB (SE) 2012-08-30 WO disclosed
EP-2491952-A1 A system for cargo delivery into the cells Cepep III AB (SE) 2012-08-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12576474-B2 Modification method of polyurethane, polyurethane, polishing pad, and modification method of polishing pad PADI2, PADI1, DUOX2 PDE3A 604/4885PTGS1 825/4885MEN1 1782/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.