Trifloxysulfuron

Trifloxysulfuron

SCHEMBL120688

COc1cc(OC)nc(NC(=O)[N-]S(=O)(=O)c2ncccc2OCC(F)(F)F)n1.[Na+]

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Trifloxysulfuron. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.39
CYP1A2 P05177 1/20 0.37
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HIF1A Q16665 1/20 0.36
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
XBP1 P17861 1/20 0.35
STAT3 P40763 1/20 0.35
MDM2 Q00987 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
MRGPRX1 Q96LB2 3/20 0.35
S1PR1 P21453 1/20 0.35
NFE2L2 Q16236 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifloxysulfuron SCHEMBL29419075 1.00 MAPT (0.40) MAPTTP53GLAGAACYP1A2
Trifloxysulfuron SCHEMBL2439050 0.93 GAA (0.47) MAPTTP53GLAGAAHTT
Trifloxysulfuron SCHEMBL64184 0.83 GAA (0.55) MAPTTP53GLAGAACYP1A2
Trifloxysulfuron SCHEMBL15449154 0.83 GAA (0.55) MAPTTP53GLAGAACYP1A2
Trifloxysulfuron SCHEMBL301007 0.82 GAA (0.54) MAPTTP53GLAGAACYP1A2
SCHEMBL5461709 0.81 GAA (0.40) MAPTTP53GLAGAACYP1A2
Trifloxysulfuron SCHEMBL14768215 0.81 GAA (0.53) MAPTTP53GLAGAACYP1A2
Trifloxysulfuron SCHEMBL19463553 0.76 GAA (0.45) MAPTTP53GLAGAAHTT
SCHEMBL1535821 0.74 GAA (0.43) MAPTTP53GLAGAACYP1A2
Trifloxysulfuron SCHEMBL14300670 0.73 GAA (0.44) MAPTTP53GLAGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3917 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12610950-B2 Method for weed control in lawn or turf DISCOVERY PURCHASER CORPORATION (US) 2026-04-28 US claimed
US-20250359550-A1 METHOD FOR WEED CONTROL IN LAWN OR TURF DISCOVERY PURCHASER CORPORATION (US) 2025-11-27 US claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
US-20250318528-A1 HERBICIDE COMPOSITION AND WEED CONTROLLING METHOD SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-10-16 US claimed
US-20250261643-A1 METHOD FOR WEED CONTROL IN LAWN OR TURF BAYER CROPSCIENCE LP 2025-08-21 US claimed
US-12185719-B2 Mixture of a folcysteine-based biostimulant and an agrotoxic substance of interest resulting in a quantitatively, qualitatively and time-related result-potentiating action as observed in an agricultural crop of a plant of interest UPL Corporation Limited (MU) 2025-01-07 US claimed
US-20240049711-A1 HERBICIDE COMPOSITION AND WEED CONTROLLING METHOD SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2024-02-15 US claimed
US-20230284618-A1 HERBICIDAL COMBINATIONS UPL CORPORATION LTD (MU) 2023-09-14 US claimed
EP-3599857-B1 HERBICIDAL MIXTURES BAYER AG (DE) 2023-08-23 EP claimed
US-20230000079-A1 COMBINATION COMPRISING A TRIKETONE HERBICIDE AND A DIPHENYLETHER HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2023-01-05 US claimed
EP-1998622-A1 HERBICIDAL COMPOSITION ISHIHARA SANGYO KAISHA, LTD. (JP) 2008-12-10 EP claimed
US-20080153704-A1 HERBICIDAL COMPOSITION KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 2008-06-26 US claimed
WO-2007119435-A1 HERBICIDAL COMPOSITION ISHIHARA SANGYO KAISHA, LTD. (JP) 2007-10-25 WO claimed
WO-2007112933-A1 REVERSE-PHASE MICROCAPSULES FOR ACTIVE INGREDIENTS, SIMPLIFIED PROCESS OF MANUFACTURE THEREOF AND COMBINED FORMULATIONS WDG-CS, ZC, EC-SC AND CX GAT MICROENCAPSULATION AG (AT) 2007-10-11 WO claimed
EP-1732390-A2 A HERBICIDAL COMBINATION Syngenta Participations AG (CH) 2006-12-20 EP claimed
JP-2006528217-A 2006-12-14 JP claimed
CN-1794911-A New safeners and their application BAYER CROPSCIENCE AG (DE) 2006-06-28 CN claimed
EP-1638397-A1 NEW SAFENERS AND THEIR APPLICATION Bayer CropScience AG (DE) 2006-03-29 EP claimed
WO-2005092101-A2 A HERBICIDAL COMBINATION SYNGENTA PARTICIPATIONS AG (CH) 2005-10-06 WO claimed
WO-2004103072-A1 NEW SAFENERS AND THEIR APPLICATION BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2004-12-02 WO claimed