SCHEMBL121452

SCHEMBL121452

O=S(=O)(Nc1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.76
CCNB1 P14635 2/20 0.76
CCNA2 P20248 2/20 0.76
CDK2 P24941 2/20 0.76
CDK7 P50613 2/20 0.76
CCNH P51946 2/20 0.76
CCNA1 P78396 2/20 0.76
FFAR4 Q5NUL3 2/20 0.76
FFAR1 O14842 1/20 0.76
KMT2A Q03164 3/20 0.70
PPARG P37231 1/20 0.65
NR3C1 P04150 1/20 0.64
PGR P06401 1/20 0.64
AR P10275 1/20 0.64
ESR2 Q92731 1/20 0.64
MAPT P10636 4/20 0.64
GAA P10253 1/20 0.64
TSHR P16473 1/20 0.62
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3762909 0.90 PGR (0.77) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL12113068 0.86 MEN1 (0.78) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL5894008 0.86 CDK1 (0.74) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL22516007 0.86 CDK1 (0.74) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL6842347 0.85 FFAR1 (0.77) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL22441723 0.85 CDK1 (0.64) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL678551 0.84 CA1 (0.65) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL27179684 0.83 LMNA (0.70) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL30926925 0.83 LMNA (0.70) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL27912548 0.83 FFAR4 (0.69) CDK1CCNB1CCNA2CDK2CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107076-A1 CDK2 INHIBITOR COMPOUNDS ALEKSIA THERAPEUTICS, INC. (US) 2026-05-21 WO disclosed
CN-102427810-A Sulfamoylbenzoic acid derivatives as TRPM8 antagonists RAQUALIA PHARMA INC 2012-04-25 CN disclosed
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
EP-2424517-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RaQualia Pharma Inc (JP) 2012-03-07 EP disclosed
WO-2010125831-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2010-11-04 WO disclosed
WO-2010125831-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2010-11-04 WO disclosed
US-7511043-B2 FXR modulators AMGEN INC. (US) 2009-03-31 US disclosed
US-7511043-B2 FXR modulators AMGEN INC. (US) 2009-03-31 US disclosed
US-7511043-B2 FXR modulators AMGEN INC. (US) 2009-03-31 US disclosed
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed
EP-1594840-A1 PIPERIDINE-BENZENESULFONAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-11-16 EP disclosed
US-20040176426-A1 FXR modulators TULARIK, INC. 2004-09-09 US disclosed
WO-2004072034-A1 PIPERIDINE-BENZENESULFONAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-08-26 WO disclosed
US-6777446-B2 FARNESOID X RECEPTOR; TREATING DISEASES ASSOCIATED WITH ABNORMALLY HIGH OR LOW CHOLESTEROL LEVELS. TULARIK, INC. 2004-08-17 US disclosed
US-20020120137-A1 Farnesoid X receptor; treating diseases associated with abnormally high or low cholesterol levels. TULARIK INC. 2002-08-29 US disclosed
WO-2002020463-A2 FXR MODULATORS TULARIK INC. (US) 2002-03-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020120137-A1 Farnesoid X receptor; treating diseases associated with abnormally high or low cholesterol levels. NR1H4, NR1H2, NR1H3 CDK1 4629/4885CCNB1 4433/4885CCNA2 4834/4885
US-20040176426-A1 FXR modulators NR1H4, CYP7A1, CYP7B1 CDK1 4495/4885CCNB1 4242/4885CCNA2 4752/4885
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof SFRP1, SOS1, FZD7 CDK1 1947/4885CCNB1 2750/4885CCNA2 3774/4885
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS TRPM8, TRPM5, TRPM6 CDK1 3126/4885CCNB1 4557/4885CCNA2 4207/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.