SCHEMBL12371251

SCHEMBL12371251

CCOCCOCCNC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.45
ALDH1A1 P00352 5/20 0.40
POLB P06746 1/20 0.34
TSHR P16473 1/20 0.33
THRB P10828 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
RECQL P46063 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16419854 1.00 KDM4E (0.45) KDM4EALDH1A1POLBTSHRTHRB
SCHEMBL22930458 1.00 KDM4E (0.45) KDM4EALDH1A1POLBTSHRTHRB
SCHEMBL20235111 1.00 KDM4E (0.45) KDM4EALDH1A1POLBTSHRTHRB
SCHEMBL5611814 0.95 KDM4E (0.41) KDM4EALDH1A1POLBTSHRTHRB
SCHEMBL22692193 0.91 KDM4E (0.40) KDM4EALDH1A1POLBTSHRTHRB
SCHEMBL9541679 0.90 KDM4E (0.45) KDM4EALDH1A1POLBMEN1KMT2A
SCHEMBL14198320 0.90 KDM4E (0.45) KDM4EALDH1A1POLBMEN1KMT2A
SCHEMBL9540608 0.90 KDM4E (0.45) KDM4EALDH1A1POLBMEN1KMT2A
SCHEMBL9972442 0.88 KDM4E (0.43) KDM4EALDH1A1POLBTSHRTHRB
SCHEMBL10330545 0.88 KDM4E (0.43) KDM4EALDH1A1POLBTSHRTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118139956-A Boron-free water-based lubricant for plastic working 汉高股份有限及两合公司 2024-06-04 CN claimed
CN-118139956-A Boron-free water-based lubricant for plastic working 汉高股份有限及两合公司 2024-06-04 CN disclosed
US-11161841-B2 Modulators of proteolysis and associated methods of use ARVINAS OPERATIONS, INC. (US) 2021-11-02 US disclosed
US-11065231-B2 Compounds and methods for the targeted degradation of interleukin-1 receptor- associated kinase 4 polypeptides ARVINAS OPERATIONS, INC. (US) 2021-07-20 US disclosed
WO-2021104120-A1 POLYETHYLENE GLYCOL CONJUGATE MEDICAMENT, PREPARATION METHOD THERFOR AND USE THEREOF 重庆阿普格雷生物科技有限公司 2021-06-03 WO disclosed
US-20190315732-A1 MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. 2019-10-17 US disclosed
US-20190151295-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE 4 POLYPEPTIDES ARVINAS OPERATIONS, INC. 2019-05-23 US disclosed
WO-2018119448-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF RAPIDLY ACCELERATED FIBROSARCOMA POLYPEPTIDES Arvinas, Inc. (US) 2018-06-28 WO disclosed
US-9561287-B2 Carrier-linked treprostinil prodrugs ASCENDIS PHARMA A/S (DK) 2017-02-07 US disclosed
US-9533056-B2 Dipeptide-based prodrug linkers for aliphatic amine-containing drugs ASCENDIS PHARMA AS (DK) 2017-01-03 US disclosed
US-20150196667-A1 STERILIZATION OF BIODEGRADABLE HYDROGELS ASCENDIS PHARMA AS (DK) 2015-07-16 US disclosed
US-8986609-B2 Sterilization of biodegradable hydrogels ASCENDIS PHARMA A/S (DK) 2015-03-24 US disclosed
US-20140296150-A1 Carrier-Linked Treprostinil Prodrugs ASCENDIS PHARMA A/S (DK) 2014-10-02 US disclosed
US-8486183-B2 Alkylamino alkyloxy (alcohol) monoalkyl ether for acid gas scrubbing process EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2013-07-16 US disclosed
US-20130030359-A1 DIPEPTIDE-BASED PRODRUG LINKERS FOR AROMATIC AMINE-CONTAINING DRUGS ASCENDIS PHARMA A/S (DK) 2013-01-31 US disclosed
US-20120253071-A1 Sterilization of biodegradable hydrogels ASCENDIS PHARMA A/S (DK) 2012-10-04 US disclosed
US-20120184489-A1 PRODRUGS COMPRISING AN INSULIN LINKER CONJUGATE SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2012-07-19 US disclosed
US-20110202328-A1 System for the determination of selective absorbent molecules through predictive correlations EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2011-08-18 US disclosed
US-20110202328-A1 System for the determination of selective absorbent molecules through predictive correlations EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2011-08-18 US disclosed
US-20100037775-A1 ALKYLAMINO ALKYLOXY (ALCOHOL) MONOALKYL ETHER FOR ACID GAS SCRUBBING PROCESS EXXON-MOBIL RESEARCH AND ENGINEERING COMPANY (US) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140296150-A1 Carrier-Linked Treprostinil Prodrugs PAH, TK1, SLC16A1 KDM4E 3700/4885ALDH1A1 1137/4885POLB 1603/4885
US-20190151295-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE 4 POLYPEPTIDES IRAK1, IRAK4, IRAK2 KDM4E 1071/4885ALDH1A1 2896/4885POLB 4307/4885
US-20100037775-A1 ALKYLAMINO ALKYLOXY (ALCOHOL) MONOALKYL ETHER FOR ACID GAS SCRUBBING PROCESS ALKBH3, ALKBH1, ALKBH2 KDM4E 721/4885ALDH1A1 276/4885POLB 1180/4885
US-20130030359-A1 DIPEPTIDE-BASED PRODRUG LINKERS FOR AROMATIC AMINE-CONTAINING DRUGS DNPEP, DDC, PEPD KDM4E 666/4885ALDH1A1 847/4885POLB 3068/4885
US-11065231-B2 Compounds and methods for the targeted degradation of interleukin-1 receptor- associated kinase 4 polypeptides IRAK1, IRAK4, IRAK2 KDM4E 1071/4885ALDH1A1 2896/4885POLB 4307/4885
US-20120184489-A1 PRODRUGS COMPRISING AN INSULIN LINKER CONJUGATE IAPP, IGF1R, INSR KDM4E 2506/4885ALDH1A1 468/4885POLB 3871/4885
US-20150196667-A1 STERILIZATION OF BIODEGRADABLE HYDROGELS USP3, USP30, USP4 KDM4E 596/4885ALDH1A1 664/4885POLB 2658/4885
US-20190315732-A1 MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE MDM2, CRBN, VHL KDM4E 2053/4885ALDH1A1 2958/4885POLB 2694/4885
US-20120253071-A1 Sterilization of biodegradable hydrogels USP3, USP30, USP4 KDM4E 596/4885ALDH1A1 664/4885POLB 2658/4885
US-11161841-B2 Modulators of proteolysis and associated methods of use MDM2, CRBN, VHL KDM4E 2053/4885ALDH1A1 2958/4885POLB 2694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.