SCHEMBL1243294

SCHEMBL1243294

CS(=O)(=O)c1ccc(NN)c(F)c1

nearest known ligand 0.71

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA1 P00915 13/20 0.71
CA2 P00918 13/20 0.71
CA9 Q16790 4/20 0.71
ALDH3A1 P30838 1/20 0.43
PTGS2 P35354 2/20 0.42
SOS1 Q07889 1/20 0.41
G6PD P11413 1/20 0.41
IDE P14735 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6514091 0.98 CA1 (0.69) CA1CA2CA9ALDH3A1PTGS2
SCHEMBL14875298 0.83 CA1 (0.49) CA1CA2CA9ALDH3A1PTGS2
SCHEMBL1244816 0.83 CA1 (1.00) CA1CA2CA9SOS1
Hydrochloric Acid SCHEMBL4735859 0.81 CA1 (0.96) CA1CA2CA9SOS1
SCHEMBL6807006 0.79 CA1 (0.44) CA1CA2CA9ALDH3A1G6PD
SCHEMBL9135441 0.79 SMN1; SMN2 (0.50) CA1CA2CA9ALDH3A1G6PD
SCHEMBL29173576 0.79 CA1 (0.45) CA1CA2CA9ALDH3A1PTGS2
Hydrochloric Acid SCHEMBL6511653 0.78 CA1 (0.43) CA1CA2CA9ALDH3A1G6PD
SCHEMBL9703261 0.78 CA2 (0.71) CA1CA2CA9
SCHEMBL9658757 0.77 KIF11 (0.46) CA1CA2CA9PTGS2G6PD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4596537-A1 NOVEL FLUORENE DERIVATIVE COMPOUND AND USE THEREOF JD Bioscience Inc. (KR) 2025-08-06 EP disclosed
WO-2024071629-A1 NOVEL FLUORENE DERIVATIVE COMPOUND AND USE THEREOF (주)제이디바이오사이언스 2024-04-04 WO disclosed
US-8822480-B2 Bicyclic heterocycle derivatives and use thereof as GPR119 modulators MERCK SHARP & DOHME CORP. (US) 2014-09-02 US disclosed
US-8822480-B2 Bicyclic heterocycle derivatives and use thereof as GPR119 modulators MERCK SHARP & DOHME CORP. (US) 2014-09-02 US disclosed
EP-2318404-B1 BICYCLIC HETEROCYCLE DERIVATIVES AND USE THEREOF AS GPR119 MODULATORS MERCK SHARP & DOHME (US) 2013-08-21 EP disclosed
EP-2318404-B1 BICYCLIC HETEROCYCLE DERIVATIVES AND USE THEREOF AS GPR119 MODULATORS MERCK SHARP & DOHME (US) 2013-08-21 EP disclosed
US-8410119-B2 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto ARENA PHARMACEUTICALS, INC. (US) 2013-04-02 US disclosed
CN-102417508-A Fused aryl and heteroaryl derivatives as modulators of metabolism and the prevention and treatment of disorders related thereto ARENA PHARM INC 2012-04-18 CN disclosed
CN-102159572-A Bicyclic heterocycle derivatives and use thereof as gpr119 modulators SCHERING CORP 2011-08-17 CN disclosed
US-20110166165-A1 BICYCLIC HETEROCYCLE DERIVATIVES AND USE THEREOF AS GPR119 MODULATORS SCHERING CORPORATION (US) 2011-07-07 US disclosed
WO-2007054668-A1 SYNTHESIS OF METHYLSULPHONYL BENZENE COMPOUNDS PEAKDALE MOLECULAR LIMITED (GB) 2007-05-18 WO disclosed
US-20070082874-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto ARENA PHARMACEUTICLAS, INC. (US) 2007-04-12 US disclosed
US-20070072844-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto ARENA PHARMACEUTICALS, INC. (US) 2007-03-29 US disclosed
US-7132426-B2 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto ARENA PHARMACEUTICALS, INC. (US) 2006-11-07 US disclosed
CN-1829718-A Fused aryl and heteroaryl derivatives as modulators of metabolism and the prevention and treatment of disorders related thereto ARENA PHARM INC (US) 2006-09-06 CN disclosed
WO-2006076455-A2 PROCESSES FOR PREPARING PYRAZOLO[3,4-D]PYRIMIDINE ETHERS ARENA PHARMACEUTICALS, INC. (US) 2006-07-20 WO disclosed
US-20060154940-A1 Processes for preparing pyrazolo[3,4-d]pyrimidine ethers ARENA PHARMACEUTICALS, INC. 2006-07-13 US disclosed
US-20060142262-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto ARENA PHARMACEUTICALS, INC. 2006-06-29 US disclosed
US-20050059650-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto ARENA PHARMACEUTICALS, INC. 2005-03-17 US disclosed
US-6727238-B2 CYCLOOXYGENASE INHIBITORS PFIZER INC. 2004-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166165-A1 BICYCLIC HETEROCYCLE DERIVATIVES AND USE THEREOF AS GPR119 MODULATORS GPR119, GPR88, GCGR CA1 4851/4885CA2 3976/4885CA9 3388/4885
US-20060142262-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto CYP7A1, CYP27A1, CYP4F3 CA1 4863/4885CA2 4651/4885CA9 4137/4885
US-20070082874-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto CYP7A1, CYP27A1, CYP4F3 CA1 4863/4885CA2 4651/4885CA9 4137/4885
US-20060154940-A1 Processes for preparing pyrazolo[3,4-d]pyrimidine ethers DPYD, GCK, PC CA1 4838/4885CA2 4616/4885CA9 4331/4885
US-20050059650-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto CYP7A1, CYP27A1, CYP4F3 CA1 4863/4885CA2 4651/4885CA9 4137/4885
US-20070072844-A1 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto CYP7A1, CYP27A1, CYP4F3 CA1 4863/4885CA2 4651/4885CA9 4137/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.