SCHEMBL12468302

SCHEMBL12468302

CS(=O)(=O)c1ccc(F)c(Br)c1F

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.39
PTGS2 P35354 11/20 0.37
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12560651 0.80 LMNA (0.44) CCR2PTGS2L3MBTL1LMNAHSD17B10
SCHEMBL4206943 0.79 TRPV4 (0.35)
SCHEMBL25728029 0.79 ALDH1A1 (0.36) LMNA
SCHEMBL6732039 0.78 L3MBTL1 (0.36) CCR2PTGS2L3MBTL1
SCHEMBL16825498 0.76 EPAS1 (0.43) CCR2LMNA
SCHEMBL28354575 0.75 CCR2 (0.39) CCR2PTGS2L3MBTL1LMNAHSD17B10
SCHEMBL8176124 0.73 CCR2 (0.38) CCR2PTGS2L3MBTL1LMNA
SCHEMBL31001623 0.73 CCR2 (0.38) CCR2PTGS2L3MBTL1LMNA
SCHEMBL16825580 0.73 CCR2 (0.33) CCR2L3MBTL1
SCHEMBL16825551 0.72 VCAM1 (0.40) CCR2LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103113-A1 PYRAZINE AND IMIDAZOLIDINE DERIVATIVES AND THEIR USES TO TREAT HEPATITIS C GILEAD PHARMASSET, LLC (US) 2012-08-02 WO disclosed