SCHEMBL12469038

SCHEMBL12469038

CN(C)CCNC(=O)c1ccc(-c2ccc(N)cc2F)c2c1C(=O)NC2.Nc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
ACKR3 P25106 1/20 0.38
BTK Q06187 9/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HTT P42858 1/20 0.38
PDGFRB P09619 2/20 0.36
KDR P35968 2/20 0.36
KIT P10721 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK14 Q16539 2/20 0.36
FGFR1 P11362 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
MAPK11 Q15759 1/20 0.35
GPR52 Q9Y2T5 1/20 0.34
RAD52 P43351 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469540 0.95 L3MBTL1 (0.40) PARP1BTKALDH1A1PRKAA2PRKAA1
SCHEMBL12469573 0.89 ALPL (0.40) BTKHTTPDGFRBKDRKIT
SCHEMBL12469508 0.88 BTK (0.40) BTKKDR
SCHEMBL12469562 0.85 BTK (0.42) BTKKDR
SCHEMBL12469581 0.84 CACNA1G (0.43) PARP1PDGFRBKDRKITFGFR1
SCHEMBL12469505 0.83 BTK (0.41) BTKKDRMAPK14
SCHEMBL12469295 0.83 SMYD2 (0.41) PDGFRBKDRKITALDH1A1
SCHEMBL12469481 0.82 ALOX5 (0.40) BTKKDRMAPK14
SCHEMBL12469512 0.82 CRBN (0.41) ACKR3BTKALDH1A1
SCHEMBL12469574 0.82 BCL3 (0.49) PARP1SMN1; SMN2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed