SCHEMBL902018

SCHEMBL902018

CC(=O)N1CCN(c2cc(-c3cccc(N)n3)cc(N)n2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.52
CKS1B P61024 1/20 0.47
SKP1 P63208 1/20 0.47
SKP2 Q13309 1/20 0.47
PIK3CA P42336 1/20 0.46
GBA1 P04062 1/20 0.43
MAP4K4 O95819 1/20 0.43
NOS1 P29475 2/20 0.42
DPP4 P27487 1/20 0.42
CASP6 P55212 1/20 0.42
GFER P55789 1/20 0.42
ABCB1 P08183 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
CNR2 P34972 1/20 0.41
PIM2 Q9P1W9 1/20 0.40
SMO Q99835 1/20 0.40
PIM1 P11309 1/20 0.40
NOS3 P29474 1/20 0.40
EIF2AK4 Q9P2K8 1/20 0.39
HDAC3 O15379 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902015 0.86 ITGB2 (0.46) NCF1CKS1BSKP1SKP2PIK3CA
SCHEMBL902069 0.83 HRH4 (0.57) HRH4
SCHEMBL12469602 0.80 HRH4 (0.45) NOS1GFERHRH4CNR2NOS3
SCHEMBL901638 0.75 PRKD3 (0.43) NOS1NOS3
SCHEMBL5469792 0.74 HRH4 (0.64) NCF1CKS1BSKP1SKP2GBA1
SCHEMBL23330166 0.74 NCF1 (0.52) NCF1CKS1BSKP1SKP2PIK3CA
SCHEMBL6619070 0.71 NOS1 (0.79) NOS1NOS3
SCHEMBL1704599 0.71 CKS1B (0.51) CKS1BSKP1SKP2PIK3CAMAP4K4
SCHEMBL27913890 0.70 GRIN2D (0.48) NCF1CKS1BSKP1SKP2MAP4K4
SCHEMBL901843 0.70 ASIC3 (0.46) NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed