SCHEMBL12499317

SCHEMBL12499317

Cn1nc(Cc2ccc(C(F)(F)F)cc2)c(C(=O)O)c1C(F)F

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.43
LMNA P02545 2/20 0.41
POLB P06746 1/20 0.41
LDHA P00338 1/20 0.40
LDHB P07195 1/20 0.40
AADAT Q8N5Z0 1/20 0.38
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
PTGER4 P35408 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
PTGER2 P43116 1/20 0.36
IDH1 O75874 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
P2RY14 Q15391 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12499380 0.86 AADAT (0.41) AADATPTGER4PTGER2MEN1KMT2A
SCHEMBL12499656 0.85 MAPT (0.43) LMNAPOLBIDH1MEN1KMT2A
SCHEMBL12499324 0.85 MAPT (0.40) LMNAPOLBLDHALDHBMEN1
SCHEMBL12498729 0.84 SRD5A2 (0.46) SRD5A2LMNAPOLBLDHALDHB
SCHEMBL12499736 0.84 SRD5A2 (0.46) SRD5A2LMNAPOLBLDHALDHB
SCHEMBL12499865 0.80 CCR2 (0.37) KDM5AKDM5BPTGER4PTGER2MEN1
SCHEMBL12498775 0.76 HCAR2 (0.42) LMNAKDM4CKDM5BPTGER4PTGER2
SCHEMBL12499839 0.73 LMNA (0.43) SRD5A2LMNAPOLBAADATIDH1
SCHEMBL12499319 0.73 KDM4E (0.43) LMNAPOLBMEN1KMT2AALDH1A1
SCHEMBL12499378 0.72 MAPT (0.40) LMNAPOLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103071-A2 COMPOUNDS AND COMPOSITIONS EISAI R&D MANAGEMENT CO., LTD. (JP) 2012-08-02 WO disclosed