SCHEMBL12499736

SCHEMBL12499736

Cn1nc(Cc2ccc(C(F)(F)F)cc2)c(C(=O)O)c1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.46
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 1/20 0.41
LDHA P00338 1/20 0.40
LDHB P07195 1/20 0.40
AADAT Q8N5Z0 1/20 0.39
KDM5A P29375 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
IDH1 O75874 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
P2RY14 Q15391 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
PTGER4 P35408 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12499378 0.88 MAPT (0.40) LMNAPOLBMEN1KMT2A
SCHEMBL12498729 0.87 SRD5A2 (0.46) SRD5A2LMNAPOLBLDHALDHB
SCHEMBL12498747 0.85 AADAT (0.43) HDAC1HDAC8AADATMEN1KMT2A
SCHEMBL12499879 0.84 MAPT (0.46) LMNAPOLBMEN1KMT2A
SCHEMBL12499317 0.84 SRD5A2 (0.43) SRD5A2LMNAPOLBHDAC1HDAC8
SCHEMBL12499826 0.83 CCR2 (0.39) KDM5AKDM5BPTGER4
SCHEMBL12499705 0.79 HCAR2 (0.42) LMNAKDM4CMEN1KMT2A
SCHEMBL2087514 0.77 PKM (0.34)
SCHEMBL12499839 0.76 LMNA (0.43) SRD5A2LMNAPOLBAADATIDH1
SCHEMBL12498738 0.73 MAPT (0.47) LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103071-A2 COMPOUNDS AND COMPOSITIONS EISAI R&D MANAGEMENT CO., LTD. (JP) 2012-08-02 WO disclosed