SCHEMBL13291365

SCHEMBL13291365

COCCOCc1nc(C)ccc1C(=O)C1C(=O)CCCC1=O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
HPD P32754 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13291364 0.83 HSD11B1 (0.32) CNR1CNR2MEN1ALDH1A1TSHR
SCHEMBL30637698 0.82 CNR1 (0.39) CNR1CNR2MEN1ALDH1A1KMT2A
SCHEMBL18323055 0.75 MEN1 (0.42) MEN1ALDH1A1TSHRKMT2AHSD17B10
SCHEMBL22443003 0.74 HPD (0.33) HPD
SCHEMBL14189387 0.73 HPD (0.41) HPD
SCHEMBL17400859 0.73 HPD (0.42) HPD
SCHEMBL20760039 0.73 MAPK1 (0.41) HPD
SCHEMBL14344337 0.72 HPD (0.44) HPDALDH1A1
SCHEMBL13744948 0.72 HPD (0.52) HPDALDH1A1KMT2A
SCHEMBL19866288 0.71 HCRTR1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 152 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144252-A1 BROMINE- OR IODINE-PARA-SUBSTITUTED [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND THEIR SALTS, AGENTS FOR PROTECTING USEFUL PLANTS OR CROP PLANTS COMPRISING THEM, METHODS FOR PRODUCING THEM AND THEIR USE AS SAFENERS BAYER AKTIENGESELLSCHAFT (DE) 2026-05-28 US disclosed
US-20260138958-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AG (DE) 2026-05-21 US disclosed
EP-4680598-A1 4-DIFLUOROMETHYL BENZAMIDES WITH HERBICIDAL ACTION Bayer Aktiengesellschaft (DE) 2026-01-21 EP disclosed
EP-4665151-A1 HERBICIDAL MIXTURES Bayer Aktiengesellschaft (DE) 2025-12-24 EP disclosed
WO-2025224076-A1 SUBSTITUTED ARYLPYRAZINES AND SALTS THEREOF, AND USE THEREOF AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2025-10-30 WO disclosed
US-20250304566-A1 CRYSTALLINE FORMS OF (5S)-3-[3-(3-CHLORO-2-FLUOROPHENOXY)-6-METHYLPYRIDAZIN-4-YL]-5-(2-CHLORO-4-METHYLBENZYL)-5,6-DIHYDRO-4H-1,2,4-OXADIAZINE BAYER AKTIENGEELLSCHAFT (DE) 2025-10-02 US disclosed
EP-4618745-A1 USE OF ISOTIANIL FOR CONTROLLING PLASMODIOPHORA BRASSICA Bayer Aktiengesellschaft (DE) 2025-09-24 EP disclosed
US-20250280829-A1 USE OF (5S)-3-[3-(3-CHLORO-2-FLUOROPHENOXY)-6-METHYLPYRIDAZIN-4-YL]-5-(2-CHLORO-4-METHYLBENZYL)-5,6-DIHYDRO-4H-1,2,4-OXADIAZINE FOR CONTROLLING UNWANTED MICROORGANISMS BAYER AKTIENGESELLSCHAFT (DE) 2025-09-11 US disclosed
EP-4384016-B1 ACTIVE COMPOUND COMBINATIONS AND FUNGICIDE COMPOSITIONS COMPRISING THOSE BAYER AG (DE) 2025-09-03 EP disclosed
EP-4605379-A1 BROMINE- OR IODINE-PARA-SUBSTITUTED [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND SALTS THEREOF, PROTECTION AGENTS COMPRISING THEM, FOR USEFUL PLANTS OR CROP PLANTS, METHODS FOR PRODUCING THEM AND USE THEREOF AS SAFENERS Bayer Aktiengesellschaft (DE) 2025-08-27 EP disclosed
WO-2022084278-A1 1-(PYRIDYL)-5-AZINYLPYRAZOLE DERIVATIVES, AND THEIR USE FOR CONTROL OF UNDESIRED PLANT GROWTH BAYER AKTIENGESELLSCHAFT (DE) 2022-04-28 WO disclosed
US-20160029629-A1 LAWN GROWTH-PROMOTING AGENT AND METHOD OF USING SAME BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-04 US disclosed
US-20160029629-A1 LAWN GROWTH-PROMOTING AGENT AND METHOD OF USING SAME BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-04 US disclosed
WO-2010063422-A1 SUBSTITUTED 1-(THIAZOLYL)- AND 1-(ISOTHIAZOLYL)PYRAZOLE-4-YL-ACETIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2010-06-10 WO disclosed
WO-2010017928-A1 HERBICIDAL COMBINATION COMPRISING DIMETHOXY-TRIAZINYL-SUBSTITUTED DIFLUOROMETHANE SULFONYANILIDES BAYER CROPSCIENCE AG (DE) 2010-02-18 WO disclosed
WO-2010017923-A2 HERBICIDAL COMBINATION WITH DIMETHOXY-TRIAZINYL-SUBSTITUTED DIFLUOROMETHANE SULFONYLANILIDES BAYER CROPSCIENCE AG (DE) 2010-02-18 WO disclosed
WO-2010017925-A2 HERBICIDAL-SAFENER-COMBINATION COMPRISING DIMETHOXYTRIAZINYL- SUBSTITUTED DIFLUORMETHANE SULFONYLANILIDES BAYER CROPSCIENCE AG (DE) 2010-02-18 WO disclosed
WO-2010017927-A2 HERBICIDAL COMBINATION COMRPISING DIMETHOXYTRIAZINYL-SUBSTITUTED DIFLUOROMETHANE SULFONYLANILIDES BAYER CROPSCIENCE AG (DE) 2010-02-18 WO disclosed
WO-2009129953-A1 2-(BENZYLSULFONYL)-OXAZOLE DERIVATIVES, CHIRAL 2- (BENZYLSULFINYL) -OXAZOLE DERIVATIVES AND 2-(BENZYLSULFANYL)-OXAZOLE DERIVATIVES, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2009-10-29 WO disclosed
WO-2009059712-A2 HOMOGENEOUS AND STORAGE-STABLE MIXTURES OF DIFFERENT ACTIVE PLANT PROTECTION AGENT GRANULE PARTICLES BAYER CROPSCIENCE AG (DE) 2009-05-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260138958-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES CBR1, CBR3, HDHD5 CNR1 374/4885CNR2 968/4885HPD 255/4885
US-20260144252-A1 BROMINE- OR IODINE-PARA-SUBSTITUTED [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND THEIR SALTS, AGENTS FOR PROTECTING USEFUL PLANTS OR CROP PLANTS COMPRISING THEM, METHODS FOR PRODUCING THEM AND THEIR USE AS SAFENERS CBR3, CBR1, CA3 CNR1 122/4885CNR2 400/4885HPD 677/4885
US-20250280829-A1 USE OF (5S)-3-[3-(3-CHLORO-2-FLUOROPHENOXY)-6-METHYLPYRIDAZIN-4-YL]-5-(2-CHLORO-4-METHYLBENZYL)-5,6-DIHYDRO-4H-1,2,4-OXADIAZINE FOR CONTROLLING UNWANTED MICROORGANISMS CYP4Z1, IL5, NT5C CNR1 994/4885CNR2 1127/4885HPD 82/4885
US-20160029629-A1 LAWN GROWTH-PROMOTING AGENT AND METHOD OF USING SAME FGF2, FGF1, MKI67 CNR1 3731/4885CNR2 2649/4885HPD 302/4885
US-20250304566-A1 CRYSTALLINE FORMS OF (5S)-3-[3-(3-CHLORO-2-FLUOROPHENOXY)-6-METHYLPYRIDAZIN-4-YL]-5-(2-CHLORO-4-METHYLBENZYL)-5,6-DIHYDRO-4H-1,2,4-OXADIAZINE CYP3A5, CYP4Z1, CASP5 CNR1 2061/4885CNR2 2214/4885HPD 47/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.