SCHEMBL134643

SCHEMBL134643

COC(=O)[C@H]1CCCCN1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
TSHR P16473 2/20 0.46
CYP2C9 P11712 1/20 0.46
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
PRCP P42785 1/20 0.40
SLC6A3 Q01959 4/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 1/20 0.40
DHFR P00374 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL40033 1.00 CYP3A4 (0.46) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
SCHEMBL40034 1.00 CYP3A4 (0.46) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
SCHEMBL15384851 0.98 CYP3A4 (0.45) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
Hydrochloric Acid SCHEMBL132158 0.98 TSHR (0.45) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
SCHEMBL17919051 0.98 CYP3A4 (0.45) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
SCHEMBL1688457 0.98 CYP3A4 (0.45) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
Hydrochloric Acid SCHEMBL134642 0.98 TSHR (0.45) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
Hydrochloric Acid SCHEMBL1899822 0.98 TSHR (0.45) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
SCHEMBL16946146 0.98 CYP3A4 (0.45) CYP3A4CYP2D6TSHRCYP2C9CYP1A2
Hydrochloric Acid SCHEMBL15206077 0.96 TSHR (0.44) CYP3A4CYP2D6TSHRCYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 130 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116735748-A Chiral purity detection method for (R) -piperidine-2-methyl formate hydrochloride 上海吉奉生物科技有限公司 2023-09-12 CN claimed
US-12624003-B2 Carboxylic acid containing indanyl compounds for the treatment of neurodegenerative diseases CELGENE CORPORATION (US) 2026-05-12 US disclosed
US-20260098060-A1 MACROCYCLIC CFTR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2026-04-09 US disclosed
EP-4267117-B1 CARBOXYLIC ACID CONTAINING INDANYL COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES CELGENE CORP (US) 2026-04-08 EP disclosed
US-20260000781-A1 FC CONJUGATES INCLUDING AN INHIBITOR OF CD73 AND USES THEREOF CIDARA THERAPEUTICS INC (US) 2026-01-01 US disclosed
EP-4587443-A1 MACROCYCLIC CFTR MODULATORS Idorsia Pharmaceuticals Ltd (CH) 2025-07-23 EP disclosed
EP-4551563-A2 FC CONJUGATES INCLUDING AN INHIBITOR OF CD73 AND USES THEREOF CIDARA THERAPEUTICS, INC. (US) 2025-05-14 EP disclosed
CN-119816487-A FC conjugates comprising CD73 inhibitors and uses thereof 奇达拉治疗公司 2025-04-11 CN disclosed
WO-2025064869-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER CIDARA THERAPEUTICS, INC. (US) 2025-03-27 WO disclosed
WO-2024213044-A1 AZACYCLO-CARBONYL-FUSED RING DERIVATIVES AND USE THEREOF Beijing Double-Crane Runchuang Technology Co., Ltd. (CN) 2024-10-17 WO disclosed
US-20100184739-A1 Modulators of ATP-Binding Cassette Transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-07-22 US disclosed
WO-2008150118-A2 NOVEL AMIDE DERIVATIVE FOR INHIBITING THE GROWTH OF CANCER CELLS HANMI PHARM. CO., LTD. (KR) 2008-12-11 WO disclosed
US-20070099934-A1 N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprotein b JANSSEN PHARMACEUTICA N.V. (BE) 2007-05-03 US disclosed
EP-1694644-A2 N-ARYL PIPERIDINE SUBSTITUTED BIPHENYLCARBOXAMIDES AS INHIBITORS OF APOLIPOPROTEIN B JANSSEN PHARMACEUTICA N.V. (BE) 2006-08-30 EP disclosed
WO-2005058824-A2 N-ARYL PIPERIDINE SUBSTITUTED BIPHENYLCARBOXAMIDES AS INHIBITORS OF APOLIPOPROTE IN B JANSSEN PHARMACEUTICA N.V. (BE) 2005-06-30 WO disclosed
CN-1093125-C Sulfamide-metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-23 CN disclosed
CN-1250445-A Sulfamide-metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2000-04-12 CN disclosed
CN-1027695-C Heterocyclic-NMDA antagonists MERRELL DOW PHARMA (US) 1995-02-22 CN disclosed
CN-1056499-A HETEROCYCLIC-NMDA ANTAGONISTS MERRELL DOW PHARMA (US) 1991-11-27 CN disclosed
US-4760065-A Trans(-)-10aR-7,8,9,10,10a,11-hexahydro-2-trifluoromethyl -13H-pyrido(1',2':3, 4)imidazo(2, 1b)quinozoline-13-one HARDTMANN GOETZ E (US) 1988-07-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100184739-A1 Modulators of ATP-Binding Cassette Transporters CFTR, ABCB1, ABCC2 CYP3A4 1862/4885CYP2D6 1732/4885TSHR 2753/4885
US-20260098060-A1 MACROCYCLIC CFTR MODULATORS CFTR, CLIC1, ARRB1 CYP3A4 857/4885CYP2D6 440/4885TSHR 701/4885
US-20070099934-A1 N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprotein b APOB, PNLIP, LIPC CYP3A4 1066/4885CYP2D6 1104/4885TSHR 2816/4885
US-12624003-B2 Carboxylic acid containing indanyl compounds for the treatment of neurodegenerative diseases S1PR5, LPAR5, S1PR2 CYP3A4 3400/4885CYP2D6 1724/4885TSHR 1869/4885
US-20260000781-A1 FC CONJUGATES INCLUDING AN INHIBITOR OF CD73 AND USES THEREOF FCGR2A, FCGR1A, FCGR3B CYP3A4 2895/4885CYP2D6 1832/4885TSHR 842/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.