SCHEMBL1347714

SCHEMBL1347714

Cc1cc(NC2CCCCC2)ccc1-c1cccc(C(N)=O)c1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FAAH O00519 6/20 0.50
TRPA1 O75762 1/20 0.50
EPHX2 P34913 1/20 0.50
FAAH2 Q6GMR7 1/20 0.50
MGLL Q99685 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
F3 P13726 1/20 0.48
HCRTR1 O43613 1/20 0.43
LRRK2 Q5S007 1/20 0.42
CSF1R P07333 1/20 0.42
FLT1 P17948 1/20 0.42
FLT3 P36888 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23609342 0.80 LMNA (0.46)
SCHEMBL1348506 0.73 OPRM1 (0.42) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL28667688 0.73 FAAH (0.66) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL16118345 0.73 FAAH (0.76) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL1786409 0.73 ALDH1A1 (0.54) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL10425208 0.72 SYK (0.51) EPHX2
SCHEMBL7113709 0.72 LRRK2 (0.50) LRRK2CSF1RFLT1FLT3
SCHEMBL1785732 0.71 OPRM1 (0.47) FAAHHDAC6
SCHEMBL31557872 0.71 PARP14 (0.61) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL31557918 0.71 ROCK2 (0.49) FAAHTRPA1EPHX2FAAH2MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063247-B2 Bicyclic aryl and heteroaryl receptor modulators PROSIDION LIMITED (GB) 2011-11-22 US claimed
US-8063247-B2 Bicyclic aryl and heteroaryl receptor modulators PROSIDION LIMITED (GB) 2011-11-22 US disclosed
US-20100267780-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2010-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100267780-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS OPRM1, OPRL1, OPRD1 FAAH 224/4885TRPA1 312/4885EPHX2 2276/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.