SCHEMBL13628514

SCHEMBL13628514

CC(C)NOC(CNc1cc(N)ccn1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 7/20 0.39
CYP2D6 P10635 1/20 0.37
ADRA1D P25100 2/20 0.36
HTR2C P28335 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
DRD2 P14416 1/20 0.36
NR3C2 P08235 1/20 0.36
FAAH O00519 3/20 0.35
NOS2 P35228 1/20 0.35
HRH4 Q9H3N8 3/20 0.34
MAPK14 Q16539 2/20 0.34
AAK1 Q2M2I8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628669 0.88 CYP2D6 (0.39) HTR7CYP2D6ADRA1DHTR2CADRA1A
SCHEMBL13628672 0.83 CYP2D6 (0.55) CYP2D6
SCHEMBL13628673 0.76 ASIC3 (0.32) NR3C2HRH4
SCHEMBL13628525 0.70 CYP2D6 (0.57) CYP2D6
SCHEMBL7459147 0.67 NOS2 (0.66) CYP2D6NOS2AAK1
SCHEMBL13628670 0.66 CYP1A2 (0.46)
SCHEMBL15102638 0.66 MAPK14 (0.42) HRH4MAPK14
SCHEMBL2642666 0.66 KCNH2 (0.41) NOS2HRH4MAPK14
SCHEMBL14224121 0.65 MTNR1A (0.51)
SCHEMBL291728 0.63 CYP2D6 (0.60) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612197-B2 Reacting a nucleophil with OH group with an electrophil to form an adduct, reacting adduct with a reagent selected from oxidizing, sulfurizing or selenizing agents to produce hydroxy protected oligonucleotide, heating to deprotect hydroxy protecting group such as 2-(2-pyridyl)aminoethoxycarbonyl The United States of America as repesented by the Secretary of the Department of Health and Human Services (US) 2009-11-03 US disclosed