SCHEMBL13639363

SCHEMBL13639363

COc1ccccc1C(=O)Oc1ccc(-c2ccc3c4c2CN(c2ccccc2OC)N4C(=O)C(C)(C)N3)c(OC)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
ESR1 P03372 1/20 0.38
IL6 P05231 6/20 0.37
MAPT P10636 5/20 0.36
HPGD P15428 2/20 0.36
XBP1 P17861 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
PLIN1 O60240 1/20 0.36
USP2 O75604 1/20 0.36
TNNI3 P19429 1/20 0.36
TNNT2 P45379 1/20 0.36
TNNC1 P63316 1/20 0.36
PLIN5 Q00G26 1/20 0.36
ABHD5 Q8WTS1 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GAA P10253 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639370 0.94 IL6 (0.38) KMT2AMEN1ESR1IL6MAPT
SCHEMBL13639336 0.91 HCRTR1 (0.37) KMT2AIL6MAPTKDM4EALDH1A1
SCHEMBL14015835 0.91 IL6 (0.39) IL6MAPTHPGDKDM4EALDH1A1
SCHEMBL14015609 0.89 DRD2 (0.36) KMT2AMEN1IL6MAPTHPGD
SCHEMBL14015605 0.89 KMT2A (0.36) KMT2AIL6MAPTHPGDNPSR1
SCHEMBL14878774 0.89 ALOX15 (0.41) KMT2AMEN1IL6MAPTHPGD
SCHEMBL14015535 0.89 ADRA1D (0.36) KMT2AMEN1IL6HPGDKDM4E
SCHEMBL13639362 0.88 HTR1A (0.37) IL6MAPTHPGDNPSR1KDM4E
SCHEMBL13639358 0.88 KMT2A (0.37) KMT2AMEN1IL6MAPTHPGD
SCHEMBL14015539 0.87 IL6 (0.37) KMT2AMEN1IL6MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1995242-B1 NOVEL 1,2,3,4-TETRAHYDROQUINOXALINE DERIVATIVE HAVING GLUCOCORTICOID RECEPTOR BINDING ACTIVITY SANTEN PHARMACEUTICAL CO LTD (JP) 2012-11-07 EP disclosed
EP-1995242-A1 NOVEL 1,2,3,4-TETRAHYDROQUINOXALINE DERIVATIVE HAVING GLUCOCORTICOID RECEPTOR BINDING ACTIVITY Santen Pharmaceutical Co., Ltd (JP) 2008-11-26 EP disclosed