SCHEMBL13680847

SCHEMBL13680847

Cc1ccc(-c2cccc(CCC=O)n2)cn1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.43
CYP2A6 P11509 1/20 0.39
IRAK4 Q9NWZ3 6/20 0.37
ELANE P08246 1/20 0.36
MAOB P27338 2/20 0.36
TRPV3 Q8NET8 1/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
WNT3A P56704 1/20 0.33
HPGDS O60760 1/20 0.33
SCN9A Q15858 1/20 0.32
GRM5 P41594 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680834 0.84 PDE10A (0.39) PDE10AIRAK4TRPV3RAB9A
SCHEMBL13680848 0.83 ADK (0.40) NPC1RAB9AKCNH2SCN9A
SCHEMBL13680846 0.83 MAPT (0.40) PDE10ACYP2A6TRPV3SCN9AGRM5
SCHEMBL13680849 0.82 SCN9A (0.43) CYP2A6SCN9AGRM5
SCHEMBL13680850 0.80 TRPV3 (0.53) TRPV3KCNH2SCN9A
SCHEMBL13680852 0.79 CYP2A6 (0.51) PDE10ACYP2A6IRAK4NPC1RAB9A
SCHEMBL3854280 0.79 MEN1 (0.50) PDE10ATRPV3RAB9AKCNH2WNT3A
SCHEMBL13680851 0.78 MAPK1 (0.43) PDE10AGRM5
SCHEMBL13680815 0.77 PDE10A (0.46) PDE10ANPC1RAB9AHRH3SCN9A
SCHEMBL13680831 0.77 PDE10A (0.37) PDE10ACYP2A6TRPV3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed