SCHEMBL13680950

SCHEMBL13680950

CC(=O)Oc1ccc(-c2nc(CCC=O)cs2)cn1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
CYP19A1 P11511 3/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
GAA P10253 1/20 0.37
MAPT P10636 5/20 0.37
TP53 P04637 4/20 0.37
POLB P06746 1/20 0.37
LMNA P02545 3/20 0.37
THRB P10828 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680959 0.86 CYP19A1 (0.53) PPARDPPARACYP19A1ALDH1A1KDM4E
SCHEMBL13680957 0.83 KDM4E (0.50) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL13680956 0.81 SHMT2 (0.40) PPARDPPARACYP19A1ALDH1A1KDM4E
SCHEMBL13680955 0.79 GAA (0.42) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL13680949 0.79 HPGDS (0.43) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL13681036 0.78 KMT2A (0.37) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL13680954 0.77 KDM4E (0.40) ALDH1A1KDM4EGAAMAPTTP53
SCHEMBL13680932 0.77 KMT2A (0.47) ALDH1A1KDM4EHPGDMAPTTP53
SCHEMBL13680953 0.77 LMNA (0.41) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL13681055 0.76 KDM4E (0.46) ALDH1A1KDM4EHPGDGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed