SCHEMBL13680959

SCHEMBL13680959

COc1ccc(-c2nc(CCC=O)cs2)cn1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.53
CYP2A6 P11509 2/20 0.42
KDM4E B2RXH2 7/20 0.41
ALDH1A1 P00352 4/20 0.41
HPGD P15428 2/20 0.41
CPT2 P23786 1/20 0.41
CPT1A P50416 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
RAB9A P51151 1/20 0.41
GAA P10253 1/20 0.40
MAPT P10636 4/20 0.39
TP53 P04637 1/20 0.39
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
F2RL3 Q96RI0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680950 0.86 PPARD (0.40) CYP19A1KDM4EALDH1A1HPGDRAB9A
SCHEMBL13680956 0.84 SHMT2 (0.40) CYP19A1KDM4EALDH1A1HPGDMAPT
SCHEMBL13680955 0.83 GAA (0.42) CYP2A6KDM4EALDH1A1HPGDCPT2
SCHEMBL13680989 0.83 KDM4E (0.39) CYP19A1KDM4EALDH1A1HPGDTDP1
SCHEMBL13680929 0.82 ALDH1A1 (0.62) KDM4EALDH1A1HPGDTDP1RAB9A
SCHEMBL13680954 0.81 KDM4E (0.40) KDM4EALDH1A1RAB9AGAAMAPT
SCHEMBL13680953 0.81 LMNA (0.41) CYP2A6KDM4EALDH1A1HPGDGAA
SCHEMBL28731211 0.80 CYP19A1 (0.56) CYP19A1CYP2A6KDM4EALDH1A1HPGD
SCHEMBL13681049 0.79 LMNA (0.38) KDM4EALDH1A1HPGDRAB9AGAA
SCHEMBL5469319 0.79 KDM4E (0.68) CYP19A1CYP2A6KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed