SCHEMBL13680975

SCHEMBL13680975

O=CCCc1ccc(-c2ccc3oc(=O)[nH]c3c2)o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.48
PDE3A Q14432 2/20 0.48
NOS1 P29475 4/20 0.43
NOS3 P29474 3/20 0.43
NOS2 P35228 3/20 0.43
NPSR1 Q6W5P4 3/20 0.43
CYP1A2 P05177 2/20 0.43
TSHR P16473 2/20 0.43
LMNA P02545 1/20 0.43
ADRA2A P08913 1/20 0.43
THPO P40225 1/20 0.43
BLM P54132 1/20 0.43
POLB P06746 1/20 0.39
OGT O15294 1/20 0.37
KMO O15229 1/20 0.36
GPR55 Q9Y2T6 1/20 0.34
MAPT P10636 4/20 0.33
GAA P10253 2/20 0.33
THRB P10828 1/20 0.33
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680976 0.81 MAPT (0.50) PDE3BPDE3ANPSR1TSHRLMNA
SCHEMBL13680991 0.76 PDE3B (0.48) PDE3BPDE3ANOS1NOS3NOS2
SCHEMBL13680971 0.75 TERT (0.44) MAPTTP53ALDH1A1KDM4EHPGD
SCHEMBL13680977 0.75 CA12 (0.40) PDE3BPDE3ANPSR1CYP1A2TSHR
SCHEMBL13680594 0.75 NOS1 (0.58) PDE3BPDE3ANOS1NOS3NOS2
SCHEMBL13680972 0.73 ALDH1A1 (0.45) PDE3BPDE3ACYP1A2LMNABLM
SCHEMBL13681029 0.72 ALDH1A1 (0.36) NPSR1CYP1A2TSHRLMNAPOLB
SCHEMBL13680904 0.72 NPC1 (0.45) MAPT
SCHEMBL13680864 0.71 ALDH1A1 (0.63) NPSR1CYP1A2TSHRPOLBMAPT
SCHEMBL13680887 0.71 ALDH1A1 (0.46) NPSR1CYP1A2TSHRLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed