SCHEMBL13680981

SCHEMBL13680981

O=CCCc1csc(-c2ccc3[nH]ncc3c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.46
AURKB Q96GD4 10/20 0.46
ROCK2 O75116 10/20 0.46
PIM1 P11309 7/20 0.46
DYRK1A Q13627 7/20 0.46
GSK3A P49840 6/20 0.46
ROCK1 Q13464 6/20 0.46
JAK2 O60674 6/20 0.46
CDK5 Q00535 5/20 0.46
CDK2 P24941 5/20 0.46
AURKA O14965 4/20 0.46
DAPK3 O43293 4/20 0.46
MARK3 P27448 3/20 0.46
LIMK1 P53667 3/20 0.46
CHEK2 O96017 2/20 0.46
PRKD2 Q9BZL6 2/20 0.46
PRKACA P17612 4/20 0.45
CLK2 P49760 4/20 0.45
CLK4 Q9HAZ1 4/20 0.45
KDR P35968 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680986 0.81 GUSB (0.45) CHEK1
SCHEMBL13681003 0.80 HRH3 (0.39) CDK5CDK5R1
SCHEMBL13680995 0.79 CDC25A (0.48) DYRK1A
SCHEMBL13680996 0.75 QPCT (0.44) QPCTQPCTL
SCHEMBL13681010 0.74 PDE3B (0.50) CDK2
SCHEMBL13680997 0.74 RAB9A (0.41) DYRK1A
SCHEMBL13680984 0.74 LMNA (0.39) CDK8TRPA1
SCHEMBL13680926 0.73 LMNA (0.56) MAPK1
SCHEMBL13680922 0.73 GFER (0.62)
SCHEMBL13680943 0.73 RAB9A (0.48) PIM1CDK5CDK5R1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed