SCHEMBL14288682

SCHEMBL14288682

Cc1cc(C)c(N2CCCCC2)c(C)c1NS(=O)(=O)c1ccc(Br)cc1OC(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALPL P05186 6/20 0.47
IDH1 O75874 1/20 0.41
HSD17B1 P14061 3/20 0.39
HSD17B2 P37059 3/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
RRM1 P23921 1/20 0.39
RRM2B Q7LG56 1/20 0.39
PPARG P37231 2/20 0.38
ADRA2A P08913 3/20 0.37
NPY5R Q15761 3/20 0.37
MCHR1 Q99705 3/20 0.37
OPRM1 P35372 1/20 0.37
CCKBR P32239 1/20 0.37
KMT2A Q03164 1/20 0.36
WDR5 P61964 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533057 0.86 ALPL (0.44) ALPLIDH1KMT2A
SCHEMBL533247 0.85 CNR2 (0.39) PPARGCCKBRKMT2AWDR5
SCHEMBL534065 0.81 PKM (0.53) ALPLKMT2AWDR5
SCHEMBL532936 0.76 MCOLN3 (0.51) ALPLKMT2A
SCHEMBL5112344 0.75 SLC40A1 (0.47)
SCHEMBL532939 0.74 EDNRA (0.43) KMT2A
SCHEMBL532999 0.74 TP53 (0.48) KMT2A
SCHEMBL532980 0.73 JAK2 (0.48) PPARGKMT2A
SCHEMBL532038 0.72 ALDH1A1 (0.54) KMT2A
SCHEMBL534062 0.72 ERAP1 (0.52) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed