SCHEMBL5325289

SCHEMBL5325289

CSc1ccc(-n2c(-c3ccc(C)cc3)cc(=O)n(Cc3ccc(C(F)(F)F)cc3)c2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.38
P2RX3 P56373 2/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
PTGS2 P35354 4/20 0.36
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
RAD51 Q06609 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5324677 0.89 RGS4 (0.46) P2RX3NPC1LMNATSHRMAPK1
SCHEMBL5323331 0.85 RGS4 (0.48) LMNARAB9AMAPTTP53POLB
SCHEMBL14622453 0.84 CYP11B1 (0.43) P2RX3NPC1LMNATSHRMAPK1
SCHEMBL5326762 0.83 LMNA (0.49) NPC1LMNAMAPK1RAB9AMAPT
SCHEMBL5328787 0.83 DNM1 (0.44) NPC1LMNAMAPTTP53POLB
SCHEMBL14624165 0.81 LMNA (0.37) P2RX3NPC1LMNATSHRMAPK1
SCHEMBL5325697 0.81 RAD51 (0.40) NPC1LMNATSHRMAPK1RAB9A
SCHEMBL5331474 0.80 PTGS2 (0.38) LMNAPTGS2MAPTPTGS1
SCHEMBL5325571 0.79 RAD51 (0.35) PTGS2RAD51HDAC4HDAC1HDAC8
SCHEMBL5328955 0.78 TP53 (0.49) MAPTTP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO claimed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed