SCHEMBL5288747

SCHEMBL5288747

COc1ccc(-n2c(-c3ccc(SC)cc3)cc(=O)n(CC#N)c2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.38
PTGS1 P23219 1/20 0.38
HTT P42858 3/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
THRB P10828 1/20 0.37
TP53 P04637 1/20 0.36
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 2/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TSHR P16473 1/20 0.35
GSK3B P49841 1/20 0.35
PTPN1 P18031 1/20 0.34
CHRNA7 P36544 2/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5281280 0.87 PTGS2 (0.39) PTGS2PTGS1KDM4ECHRNA7
SCHEMBL14624155 0.85 KDM4E (0.33) PTGS2PTGS1HTTMAPTKDM4E
SCHEMBL5288324 0.84 L3MBTL1 (0.36) PTGS2MAPTKDM4EALDH1A1MEN1
SCHEMBL5323331 0.81 RGS4 (0.48) HTTMAPTKDM4ETP53ALDH1A1
SCHEMBL14624160 0.77 HTT (0.35) PTGS2PTGS1HTTTHRBLMNA
SCHEMBL5296183 0.75 POLB (0.34) PTGS2PTGS1HTTKDM4ETHRB
SCHEMBL5328955 0.75 TP53 (0.49) MAPTTHRBTP53KMT2A
SCHEMBL5294487 0.74 POLB (0.39) PTGS2PTGS1HTTMAPTKDM4E
SCHEMBL5325697 0.74 RAD51 (0.40) PTGS2PTGS1HTTTHRBLMNA
SCHEMBL5280436 0.73 POLB (0.37) PTGS2PTGS1HTTMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO claimed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed