SCHEMBL14720407

SCHEMBL14720407

O=C(O)N1CC[C@@H](CN(C(=O)c2ccc(Br)cc2)c2cnccn2)C1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.39
LMNA P02545 1/20 0.36
ACHE P22303 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
GRIN2B Q13224 1/20 0.35
VNN1 O95497 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
THRB P10828 2/20 0.34
CHRM2 P08172 1/20 0.34
MAPK14 Q16539 1/20 0.34
OPRD1 P41143 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PTGIR P43119 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720449 0.85 CHRM3 (0.52) CHRM3LMNAACHECYP3A4CYP2D6
SCHEMBL14720297 0.77 LIMK2 (0.48) CHRM3ACHECHRM2OPRD1KMT2A
SCHEMBL14720344 0.75 OPRM1 (0.42) OPRD1KDM4E
SCHEMBL14720668 0.74 OPRD1 (0.39) CHRM3HRH3THRBCHRM2OPRD1
SCHEMBL14720494 0.74 LMNA (0.33) CHRM3LMNAPTGIR
SCHEMBL14720201 0.73 HDAC1 (0.52) CHRM3CHRM2KMT2A
SCHEMBL14731355 0.73 FASN (0.58)
SCHEMBL14720130 0.67 CHIT1 (0.52) LMNAKMT2AKDM4E
SCHEMBL20549605 0.67 RAB9A (0.42) LMNAKMT2A
SCHEMBL20893533 0.67 POLB (0.53) CYP3A4CYP2D6CYP2C9KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013028445-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO disclosed