SCHEMBL14722283

SCHEMBL14722283

COc1cccn(Cc2ccc(C=C3CCN(C4CCC4)CC3)cc2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
HCRTR2 O43614 8/20 0.39
HCRTR1 O43613 7/20 0.37
MAPT P10636 2/20 0.37
CNR1 P21554 3/20 0.37
CNR2 P34972 3/20 0.37
ALDH1A1 P00352 2/20 0.36
ABCB1 P08183 1/20 0.36
ACHE P22303 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14721926 0.87 POLB (0.39) MAPTCNR1CNR2ALDH1A1KDM4E
SCHEMBL14722952 0.83 TRPV6 (0.38) HCRTR2HCRTR1MAPTCNR1CNR2
SCHEMBL14722534 0.82 LMNA (0.46) LMNAHCRTR2HCRTR1MAPTALDH1A1
SCHEMBL14722538 0.81 POLB (0.36)
SCHEMBL14723108 0.78 VEGFA (0.46) LMNAMAPTABCB1TP53
SCHEMBL14721908 0.77 HRH3 (0.36) ACHE
SCHEMBL14720875 0.74 FKBP1A (0.38)
SCHEMBL14720876 0.74 FKBP1A (0.38)
SCHEMBL14731087 0.74 KDM4E (0.42) LMNACNR2ALDH1A1KDM4E
SCHEMBL14720643 0.73 OPRM1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO claimed