Denaverine

Denaverine

SCHEMBL147346

CCC(CC)COC(C(=O)OCCN(C)C)(c1ccccc1)c1ccccc1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.52
CYP2D6 P10635 3/20 0.52
ALDH1A1 P00352 1/20 0.49
CHRM1 P11229 6/20 0.48
CHRM2 P08172 5/20 0.48
CHRM3 P20309 5/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 3/20 0.47
LMNA P02545 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
GAA P10253 1/20 0.47
CHRM4 P08173 3/20 0.46
CHRM5 P08912 1/20 0.46
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
SCN1A P35498 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Denaverine SCHEMBL9569397 0.99 CYP3A4 (0.54) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
Dimenoxadol SCHEMBL25993 0.85 CYP3A4 (0.68) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
Dimenoxadol SCHEMBL79044 0.84 CYP3A4 (0.70) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
Dimenoxadol SCHEMBL2886211 0.84 CYP3A4 (0.70) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
Dimenoxadol SCHEMBL5854258 0.83 CYP3A4 (0.69) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
SCHEMBL29519508 0.82 CYP3A4 (0.46) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
Dimenoxadol SCHEMBL2204879 0.82 CYP3A4 (0.67) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
Pargeverine SCHEMBL2111437 0.80 CYP3A4 (0.51) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
Pargeverine SCHEMBL30728632 0.79 CYP3A4 (0.53) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2
SCHEMBL9047924 0.78 LMNA (0.42) CYP3A4CYP2D6ALDH1A1CHRM1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 105 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20240074995-A1 METHODS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH AN ABNORMAL INFLAMMATORY RESPONSES FIRST WAVE BIO, INC. 2024-03-07 US disclosed
US-11793777-B2 Methods and compositions for treating conditions associated with an abnormal inflammatory response FIRST WAVE BIO, INC. (US) 2023-10-24 US disclosed
US-11744812-B2 Methods of treatment FIRST WAVE BIO, INC. (US) 2023-09-05 US disclosed
US-20230201143-A1 METHODS OF TREATMENT FIRST WAVE BIO, INC. 2023-06-29 US disclosed
WO-2023118074-A1 COMPRESSIBLE AND FREE FLOWING CO-PROCESSED MESOPOROUS SILICA UNIVERZA V LJUBLJANI (SI) 2023-06-29 WO disclosed
US-20230190684-A1 METHODS OF TREATING COVID-19 WITH A NICLOSAMIDE COMPOUND FIRST WAVE BIO, INC. 2023-06-22 US disclosed
US-20230102999-A1 DEUTERATED NICLOSAMIDE FIRST WAVE BIO, INC. 2023-03-30 US disclosed
US-6680047-B2 FOR USE IN ULTRASOUND IMAGING, CONTRAST AGENTS AMERSHAM HEALTH AS (NO) 2004-01-20 US disclosed
US-20020102217-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 US disclosed
US-20020102215-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 US disclosed
US-6331289-B1 ULTRASOUND CONTRAST AGENTS, SUSPENSION IN AQUEOUS CARRIER LIQUID OF A REPORTER COMPRISING GAS-CONTAINING OR GAS-GENERATING MATERIAL, AGENT CAPABLE OF FORMING AT LEAST TWO TYPES OF BINDING PAIRS WITH TARGET; REPORTER BEING CONJUGATED NYCOMED IMAGING AS (NO) 2001-12-18 US disclosed
US-6264917-B1 MIXTURE OF GAS FILLED MICROBUBBLES AND RELEASING AGENT NYCOMED IMAGING AS (NO) 2001-07-24 US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 US disclosed
EP-0537608-A2 Process for the technical preparation of 2,2-diphenyl-2-(2-ethyl-butoxy)acetic acid, 2-dimethyl-amino-ethyl ester, hydrochloride APOGEPHA ARZNEIMITTEL GmbH (DE) 1993-04-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240074995-A1 METHODS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH AN ABNORMAL INFLAMMATORY RESPONSES FH, CS, ECHS1 CYP3A4 1499/4885CYP2D6 953/4885ALDH1A1 2174/4885
US-20230190684-A1 METHODS OF TREATING COVID-19 WITH A NICLOSAMIDE COMPOUND ACE2, ACE, MME CYP3A4 141/4885CYP2D6 179/4885ALDH1A1 3497/4885
US-11744812-B2 Methods of treatment ACE2, ACE, SI CYP3A4 212/4885CYP2D6 239/4885ALDH1A1 3977/4885
US-20230201143-A1 METHODS OF TREATMENT ACE2, ACE, SI CYP3A4 209/4885CYP2D6 259/4885ALDH1A1 3889/4885
US-20230102999-A1 DEUTERATED NICLOSAMIDE FH, IDH2, ECHS1 CYP3A4 1035/4885CYP2D6 243/4885ALDH1A1 2305/4885
US-11793777-B2 Methods and compositions for treating conditions associated with an abnormal inflammatory response FH, CS, ECHS1 CYP3A4 1393/4885CYP2D6 865/4885ALDH1A1 2230/4885
US-20020102215-A1 Diagnostic/therapeutic agents BID, FUS, FABP1 CYP3A4 4863/4885CYP2D6 4855/4885ALDH1A1 4459/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.