Pantoprazole

Pantoprazole

SCHEMBL1476069

COc1ccnc(C[S+]([O-])c2nc3cc(OC(F)F)ccc3[nH]2)c1OC.O.O.[NaH]

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Pantoprazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A known ✓ P20648 14/20 0.52
ATP4B known ✓ P51164 14/20 0.52
ADRA1A known ✓ P35348 1/20 0.52
CYP2C9 P11712 2/20 0.52
KDM4E B2RXH2 1/20 0.52
SLC22A2 O15244 1/20 0.52
DDAH1 O94760 1/20 0.52
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
ABCB1 P08183 1/20 0.52
CYP3A4 P08684 1/20 0.52
MAPT P10636 1/20 0.52
HPGD P15428 1/20 0.52
ALOX15 P16050 1/20 0.52
FASN P49327 1/20 0.52
SLC47A2 Q86VL8 1/20 0.52
SLC47A1 Q96FL8 1/20 0.52
ABCG2 Q9UNQ0 1/20 0.52
ATP1A1 P05023 7/20 0.44
ATP1B1 P05026 7/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pantoprazole SCHEMBL21986309 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL1477291 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL27913225 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL1476428 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL3542 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL6262319 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL5795111 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL3179774 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL4199906 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL1560742 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114028359-B Pantoprazole quick-release capsule and preparation method thereof 厦门恩成制药有限公司 2023-03-17 CN claimed
CN-114028359-A Pantoprazole quick-release capsule and preparation method thereof 厦门恩成制药有限公司 2022-02-11 CN claimed
EP-1572680-A2 SOLID STATES OF PANTOPRAZOLE SODIUM, KNOWN PANTOPRAZOLE SODIUM HYDRATES, PROCESSES FOR THEIR PREPARATION. EVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2005-09-14 EP claimed
US-20040177804-A1 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 2004-09-16 US claimed
WO-2004056804-A2 SOLID STATES OF PANTOPRAZOLE SODIUM, PROCESSES FOR PREPARING THEM AND PROCESSES FOR PREPARING KNOWN PANTOPRAZOLE SODIUM HYDRATES TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2004-07-08 WO claimed
CN-114028359-B Pantoprazole quick-release capsule and preparation method thereof 厦门恩成制药有限公司 2023-03-17 CN disclosed
CN-114028359-A Pantoprazole quick-release capsule and preparation method thereof 厦门恩成制药有限公司 2022-02-11 CN disclosed
EP-3397630-B1 PROCESS FOR THE PREPARATION OF PANTOPRAZOLE SODIUM SESQUIHYDRATE KRKA TOVARNA ZDRAVIL D D NOVO MESTO (SI) 2021-05-26 EP disclosed
EP-3397630-A1 PROCESS FOR THE PREPARATION OF PANTOPRAZOLE SODIUM SESQUIHYDRATE KRKA, tovarna zdravil, d.d., Novo mesto (SI) 2018-11-07 EP disclosed
WO-2017114898-A1 PROCESS FOR THE PREPARATION OF PANTOPRAZOLE SODIUM SESQUIHYDRATE KRKA, TOVARNA ZDRAVIL, D.D., NOVO MESTO (SI) 2017-07-06 WO disclosed
EP-3187494-A1 PROCESS FOR THE PREPARATION OF PANTOPRAZOLE SODIUM SESQUIHYDRATE KRKA, tovarna zdravil, d.d., Novo mesto (SI) 2017-07-05 EP disclosed
CN-104257616-A Pantoprazole sodium freeze-dried powder injection and preparation method thereof NORTHEAST PHARMACEUTICAL GROUP SHENYANG NO 1 PHARMACEUTICAL CO LTD 2015-01-07 CN disclosed
US-7915423-B2 Dissolving pantoprazole and sodium hydroxide in 2-propanol, tetrahydrofuran, acetonitrile, methanol, ethanol, water, mixtures of sec-butanol and dichloromethane, or ethyl acetate diluent, crystallizing pantoprazole sodium sesquihydrate, isolating TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 2011-03-29 US disclosed
US-7507829-B2 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates TEVA PHARMACEUTICALS INDUSTRIES, LTD (IL) 2009-03-24 US disclosed
US-20080132707-A1 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates TEVA PHARMACEUTICALS USA, INC. FOR BARBADOS. 2008-06-05 US disclosed
EP-1795530-A1 Process for preparing known pantoprazole sodium sesquihydrate Teva Pharmaceutical Industries Limited (IL) 2007-06-13 EP disclosed
EP-1572680-A2 SOLID STATES OF PANTOPRAZOLE SODIUM, KNOWN PANTOPRAZOLE SODIUM HYDRATES, PROCESSES FOR THEIR PREPARATION. EVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2005-09-14 EP disclosed
US-20040177804-A1 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 2004-09-16 US disclosed
WO-2004056804-A2 SOLID STATES OF PANTOPRAZOLE SODIUM, PROCESSES FOR PREPARING THEM AND PROCESSES FOR PREPARING KNOWN PANTOPRAZOLE SODIUM HYDRATES TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2004-07-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132707-A1 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates PROC, PRKD3, PDXK ATP4A 702/4885ATP4B 409/4885ADRA1A 2910/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.