Pantoprazole

Pantoprazole

SCHEMBL1476428

COc1ccnc(C[S+]([O-])c2nc3cc(OC(F)F)ccc3[nH]2)c1OC.O.[NaH]

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Pantoprazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A known ✓ P20648 14/20 0.52
ATP4B known ✓ P51164 14/20 0.52
ADRA1A known ✓ P35348 1/20 0.52
CYP2C9 P11712 2/20 0.52
KDM4E B2RXH2 1/20 0.52
SLC22A2 O15244 1/20 0.52
DDAH1 O94760 1/20 0.52
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
ABCB1 P08183 1/20 0.52
CYP3A4 P08684 1/20 0.52
MAPT P10636 1/20 0.52
HPGD P15428 1/20 0.52
ALOX15 P16050 1/20 0.52
FASN P49327 1/20 0.52
SLC47A2 Q86VL8 1/20 0.52
SLC47A1 Q96FL8 1/20 0.52
ABCG2 Q9UNQ0 1/20 0.52
ATP1A1 P05023 7/20 0.44
ATP1B1 P05026 7/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pantoprazole SCHEMBL1476069 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL21986309 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL1477291 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL27913225 1.00 ATP4A (0.52) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL3542 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL6262319 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL5795111 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL3179774 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL4199906 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2
Pantoprazole SCHEMBL1560742 0.99 ATP4A (0.53) ATP4AATP4BCYP2C9KDM4ESLC22A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 128 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118267481-A Construction and application of mRNA nano delivery system with environment adaptability and cooperative regulation 浙江大学 2024-07-02 CN claimed
CN-114028359-B Pantoprazole quick-release capsule and preparation method thereof 厦门恩成制药有限公司 2023-03-17 CN claimed
CN-114028359-A Pantoprazole quick-release capsule and preparation method thereof 厦门恩成制药有限公司 2022-02-11 CN claimed
CN-107550871-B Freeze-dried composition containing pantoprazole sodium 杭州中美华东制药有限公司 2020-07-21 CN claimed
CN-111057044-A Preparation method of single crystal form of pantoprazole sodium sesquihydrate 北京民康百草医药科技有限公司 2020-04-24 CN claimed
CN-107550871-A A kind of freeze-dried composition containing Pantoprazole Sodium 杭州中美华东制药有限公司 2018-01-09 CN claimed
CN-104257616-B A kind of freeze-dried powder injection of pantoprazole sodium and preparation method thereof 东北制药集团沈阳第制药有限公司 2017-07-14 CN claimed
CN-105111189-A Pantoprazole sodium compound monohydrate sphaerocrystal and preparation method thereof UNIV TIANJIN 2015-12-02 CN claimed
CN-104257616-A Pantoprazole sodium freeze-dried powder injection and preparation method thereof NORTHEAST PHARMACEUTICAL GROUP SHENYANG NO 1 PHARMACEUTICAL CO LTD 2015-01-07 CN claimed
US-20100016605-A1 Process CIPLA LIMITED (IN) 2010-01-21 US claimed
US-7507829-B2 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates TEVA PHARMACEUTICALS INDUSTRIES, LTD (IL) 2009-03-24 US claimed
EP-1901719-A2 BENZIMIDAZOLE FORMULATION Nycomed Danmark ApS (DK) 2008-03-26 EP claimed
EP-1895990-A2 FORMULATIONS CONTAINING PANTOPRAZOLE FREE ACID AND ITS SALTS Combino Pharm, S.L. (ES) 2008-03-12 EP claimed
WO-2007029124-A2 FORMULATIONS CONTAINING PANTOPRAZOLE FREE ACID AND ITS SALTS COMBINO PHARM, S.L. (US) 2007-03-15 WO claimed
US-20070020334-A1 Benzimidazole formulation TAKEDA PHARMA A/S (DK) 2007-01-25 US claimed
WO-2006105798-A2 BENZIMIDAZOLE FORMULATION NYCOMED DANMARK APS (DK) 2006-10-12 WO claimed
WO-2006064249-A2 PROCESS FOR THE PREPARATION OF PANTOPRAZOLE SODIUM CIPLA LIMITED (IN) 2006-06-22 WO claimed
EP-1572680-A2 SOLID STATES OF PANTOPRAZOLE SODIUM, KNOWN PANTOPRAZOLE SODIUM HYDRATES, PROCESSES FOR THEIR PREPARATION. EVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2005-09-14 EP claimed
US-20040177804-A1 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 2004-09-16 US claimed
WO-2004056804-A2 SOLID STATES OF PANTOPRAZOLE SODIUM, PROCESSES FOR PREPARING THEM AND PROCESSES FOR PREPARING KNOWN PANTOPRAZOLE SODIUM HYDRATES TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2004-07-08 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016605-A1 Process MPST, HPD, POR ATP4A 1157/4885ATP4B 598/4885ADRA1A 3906/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.