Pivhydrazine

Pivhydrazine

SCHEMBL149084

CC(C)(C)C(=O)NNCc1ccccc1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.57
RIPK1 Q13546 1/20 0.53
POLB P06746 2/20 0.51
LMNA P02545 4/20 0.48
CYP1A2 P05177 2/20 0.48
PTGS2 P35354 1/20 0.48
RECQL P46063 1/20 0.47
MMP8 P22894 1/20 0.47
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
CYP2C9 P11712 2/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 1/20 0.46
ALOX12 P18054 1/20 0.46
CYP2C19 P33261 1/20 0.46
OPRK1 P41145 1/20 0.45
ESRRG P62508 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pivhydrazine SCHEMBL9551290 0.98 SMN1; SMN2 (0.55) SMN1; SMN2RIPK1POLBLMNACYP1A2
Pivhydrazine SCHEMBL1933734 0.89 SMN1; SMN2 (0.48) SMN1; SMN2RIPK1POLBLMNACYP1A2
SCHEMBL1653407 0.82 CYP1A2 (0.54) SMN1; SMN2LMNACYP1A2PTGS2RAB9A
SCHEMBL24847549 0.82 CYP1A2 (0.54) SMN1; SMN2LMNACYP1A2PTGS2RAB9A
SCHEMBL1516186 0.81 RIPK1 (0.71) SMN1; SMN2RIPK1POLBLMNACYP1A2
SCHEMBL9551367 0.80 RECQL (0.48) SMN1; SMN2RIPK1POLBLMNACYP1A2
SCHEMBL9551354 0.79 ANPEP (0.49) SMN1; SMN2MMP8
SCHEMBL8843180 0.79 LMNA (0.59) SMN1; SMN2RIPK1POLBLMNACYP1A2
SCHEMBL4418820 0.79 LMNA (0.51) SMN1; SMN2LMNACYP1A2PTGS2RAB9A
SCHEMBL10480353 0.78 SMN1; SMN2 (0.75) SMN1; SMN2RIPK1POLBLMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 431 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250339403-A1 Tryptamine Formulations and Uses Thereof Natural MedTech Pty Ltd (AU) 2025-11-06 US claimed
EP-4618981-A1 COMBINATIONS OF MONOAMINE OXIDASE INHIBITORS AND SEROTONIN RECEPTOR AGONISTS AND THEIR THERAPEUTIC USE Remedi, Inc. (US) 2025-09-24 EP claimed
EP-4615444-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural Medtech Pty Ltd (AU) 2025-09-17 EP claimed
WO-2025151884-A1 USE OF GLYCOSAMINOGLYCAN SULFATED POLYSACCHARIDES SUCH AS SODIUM PENTOSAN POLYSULFATE IN COMBINATION WITH PERMEATION AGENTS TO TREAT ALZHEIMER'S DISEASE PARSONS C LOWELL (US) 2025-07-17 WO claimed
EP-4479032-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS Sage Therapeutics, Inc. (US) 2024-12-25 EP claimed
WO-2024108195-A1 COMBINATIONS OF MONOAMINE OXIDASE INHIBITORS AND SEROTONIN RECEPTOR AGONISTS AND THEIR THERAPEUTIC USE REMEDI, INC. (US) 2024-05-23 WO claimed
WO-2024098098-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural MedTech Pty Ltd (AU) 2024-05-16 WO claimed
US-20230381168-A1 ADJUNCTIVE THERAPY FOR DEPRESSION ANEUROTECH BV (BE) 2023-11-30 US claimed
WO-2023158668-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS SAGE THERAPEUTICS, INC. (US) 2023-08-24 WO claimed
WO-2023159035-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS SAGE THERAPEUTICS, INC. (US) 2023-08-24 WO claimed
US-20200038420-A1 AMINOSTEROL COMPOSITIONS AND METHODS OF USING THE SAME FOR TREATING DEPRESSION ENTERIN, INC. (US) 2020-02-06 US claimed
WO-2018200381-A1 PHARMACEUTICAL COMPOSITION COMPRISING TRYPTOPHAN AND PHYLLOKININ DERIVATIVE FOR USE IN TREATING PSYCHIATRIC AND PSYCHOLOGICAL CONDITIONS TEMPLE OTORONGO LLC (US) 2018-11-01 WO claimed
EP-2506717-B1 METHOD OF USING DOPAMINE REUPTAKE INHIBITORS AND THEIR ANALOGS FOR TREATING DIABETES SYMPTOMS AND DELAYING OR PREVENTING DIABETES-ASSOCIATED PATHOLOGIC CONDITIONS PERKINELMER INC (US) 2015-03-25 EP claimed
US-20130131127-A1 METHOD OF USING DOPAMINE REUPTAKE INHIBITORS AND THEIR ANALOGS FOR TREATING DIABETES SYMPTOMS AND DELAYING OR PREVENTING DIABETES-ASSOCIATED PATHOLOGIC CONDITIONS CALIPER LIFE SCIENCES, INC. 2013-05-23 US claimed
CN-102791134-A Method of using dopamine reuptake inhibitors and their analogs for treating diabetes symptoms and delaying or preventing diabetes-associated pathologic conditions PERKINELMER INC 2012-11-21 CN claimed
EP-2506717-A1 METHOD OF USING DOPAMINE REUPTAKE INHIBITORS AND THEIR ANALOGS FOR TREATING DIABETES SYMPTOMS AND DELAYING OR PREVENTING DIABETES-ASSOCIATED PATHOLOGIC CONDITIONS PerkinElmer, Inc. (US) 2012-10-10 EP claimed
WO-2011138142-A1 COMPOSITIONS AND USE OF SULFASALAZINE ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (EPFL) (CH) 2011-11-10 WO claimed
WO-2011069051-A1 METHOD OF USING DOPAMINE REUPTAKE INHIBITORS AND THEIR ANALOGS FOR TREATING DIABETES SYMPTOMS AND DELAYING OR PREVENTING DIABETES-ASSOCIATED PATHOLOGIC CONDITIONS CALIPER LIFE SCIENCES, INC. (US) 2011-06-09 WO claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130131127-A1 METHOD OF USING DOPAMINE REUPTAKE INHIBITORS AND THEIR ANALOGS FOR TREATING DIABETES SYMPTOMS AND DELAYING OR PREVENTING DIABETES-ASSOCIATED PATHOLOGIC CONDITIONS SLC6A3, SLC6A2, DBH SMN1; SMN2 405/4885RIPK1 2167/4885POLB 3904/4885
US-20200038420-A1 AMINOSTEROL COMPOSITIONS AND METHODS OF USING THE SAME FOR TREATING DEPRESSION HSD17B7, CYP17A1, HSD17B2 SMN1; SMN2 3529/4885RIPK1 4730/4885POLB 2765/4885
US-20230381168-A1 ADJUNCTIVE THERAPY FOR DEPRESSION HTR2A, HTR3B, HTR5A SMN1; SMN2 4119/4885RIPK1 4041/4885POLB 2605/4885
US-20250339403-A1 Tryptamine Formulations and Uses Thereof MAOA, MAOB, TPH1 SMN1; SMN2 1359/4885RIPK1 4522/4885POLB 3450/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.