SCHEMBL14965688

SCHEMBL14965688

O=C(c1cccc(C(F)(F)F)c1)N1CCC(N2CCOc3nc([N+](=O)[O-])cn3CC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RBP4 P02753 1/20 0.45
HSD11B1 P28845 2/20 0.43
LMNA P02545 2/20 0.43
POLB P06746 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MGLL Q99685 1/20 0.42
SERPINE1 P05121 1/20 0.42
L3MBTL3 Q96JM7 5/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
ACACB O00763 1/20 0.39
ACACA Q13085 1/20 0.39
SCN9A Q15858 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
L3MBTL4 Q8NA19 1/20 0.39
JAK2 O60674 2/20 0.38
JAK1 P23458 2/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965802 0.90 L3MBTL3 (0.43) HSD11B1LMNAHPGDMGLLL3MBTL3
SCHEMBL14965608 0.83 CHRM1 (0.48) HSD11B1MGLLL3MBTL3L3MBTL1SCN9A
SCHEMBL14965860 0.76 ALDH1A1 (0.52) ALDH1A1HPGDKDM4EL3MBTL3L3MBTL1
SCHEMBL14965829 0.76 ALDH1A1 (0.39) LMNAALDH1A1KDM4EMAPT
SCHEMBL14966212 0.75 HSD11B1 (0.44) HSD11B1ALDH1A1KDM4EMGLL
SCHEMBL14965836 0.75 MCHR1 (0.41) ALDH1A1
SCHEMBL14965755 0.74 EPHX2 (0.50) POLBJAK2JAK1
SCHEMBL14965864 0.73 ITGB3 (0.39) LMNAALDH1A1KDM4E
SCHEMBL14966196 0.73 ALDH1A1 (0.49) LMNAPOLBALDH1A1HPGDKDM4E
SCHEMBL14965968 0.73 LMNA (0.48) LMNAALDH1A1KDM4ESERPINE1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed