SCHEMBL1502471

SCHEMBL1502471

NC(=O)C12CCC(CC1)CC2

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.39
TDP1 Q9NUW8 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30363546 0.97 PKM (0.37) PKM
SCHEMBL218350 0.86 ALDH1A1 (0.40) PKMTDP1ALDH1A1HTTNPSR1
SCHEMBL9951769 0.79 ALDH1A1 (0.36) PKMALDH1A1HTTNPSR1
SCHEMBL20910305 0.78 PKM (0.48) PKMTDP1ALDH1A1
SCHEMBL587339 0.74 FFAR3 (0.35) PKMTDP1ALDH1A1HTTNPSR1
SCHEMBL15514232 0.74 ALDH1A1 (0.31) ALDH1A1HTTNPSR1
SCHEMBL22941948 0.74 PKM (0.32) PKM
SCHEMBL25041122 0.73 ALDH1A1 (0.33) ALDH1A1HTT
SCHEMBL20721222 0.72 ALDH1A1 (0.33) ALDH1A1HTTNPSR1
SCHEMBL7723088 0.72 ALDH1A1 (0.33) ALDH1A1HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4423075-B1 CCR6 RECEPTOR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2026-03-25 EP claimed
CN-115667259-B Fused ring compounds for inhibiting H-PGDS 佐藤制药株式会社 2025-06-17 CN claimed
EP-4423075-A1 CCR6 RECEPTOR MODULATORS Idorsia Pharmaceuticals Ltd (CH) 2024-09-04 EP claimed
CN-118401522-A Azaindole derivatives inhibiting H-PGDS 佐藤制药株式会社 2024-07-26 CN claimed
EP-4175949-A1 METHODS AND COMPOSITIONS FOR TARGETING TREGS USING CCR8 INHIBITORS Nanjing Immunophage Biotech Co., Ltd. (CN) 2023-05-10 EP claimed
WO-2023073082-A1 CCR6 RECEPTOR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2023-05-04 WO claimed
CN-115989223-A Methods and compositions for targeting Tregs using CCR8 inhibitors 南京艾美斐生物医药科技有限公司 2023-04-18 CN claimed
CN-115667259-A Condensed ring compounds for inhibiting H-PGDS 佐藤制药株式会社 2023-01-31 CN claimed
US-20260049159-A1 ANTIBODY-ALK5 INHIBITOR CONJUGATES AND THEIR USES SYNTHIS THERAPEUTICS, INC. (US) 2026-02-19 US disclosed
US-12473377-B2 Antibody-ALK5 inhibitor conjugates and their uses SYNTHIS THERAPEUTICS, INC. (US) 2025-11-18 US disclosed
CN-115667259-B Fused ring compounds for inhibiting H-PGDS 佐藤制药株式会社 2025-06-17 CN disclosed
US-20250074906-A1 AZAINDOLE DERIVATIVE THAT INHIBITS H-PGDS SATO PHARMACEUTICAL CO., LTD. (JP) 2025-03-06 US disclosed
WO-2025024726-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE KINNATE BIOPHARMA INC. (US) 2025-01-30 WO disclosed
CN-118666869-A Bridged ring compounds, pharmaceutical composition and application thereof 上海湃隆生物科技有限公司 2024-09-20 CN disclosed
EP-1581515-A1 TRIAZOLE DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE-1 Merck & Co., Inc. (US) 2005-10-05 EP disclosed
US-20050154038-A1 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1 MERCK SHARP & DOHME LLC 2005-07-14 US disclosed
US-6849636-B2 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1 MERCK & CO., INC. (US) 2005-02-01 US disclosed
WO-2004058730-A2 TRIAZOLE DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE-1 MERCK & CO., INC. (US) 2004-07-15 WO disclosed
WO-2004058741-A1 TRIAZOLE DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE-1 MERCK & CO., INC. (US) 2004-07-15 WO disclosed
US-20040133011-A1 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1 MERCK SHARP & DOHME LLC 2004-07-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12473377-B2 Antibody-ALK5 inhibitor conjugates and their uses ALK, ALKBH5, ALKBH3 PKM 4151/4885TDP1 2116/4885ALDH1A1 346/4885
US-20250074906-A1 AZAINDOLE DERIVATIVE THAT INHIBITS H-PGDS HPGDS, PTGIS, HPGD PKM 2796/4885TDP1 4241/4885ALDH1A1 780/4885
US-20050154038-A1 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1 HSD11B1, HSD17B1, HSD3B1 PKM 1889/4885TDP1 691/4885ALDH1A1 145/4885
US-20260049159-A1 ANTIBODY-ALK5 INHIBITOR CONJUGATES AND THEIR USES ALK, CD2, TGFBR2 PKM 2514/4885TDP1 3038/4885ALDH1A1 586/4885
US-20040133011-A1 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1 HSD11B1, HSD17B1, HSD3B1 PKM 1910/4885TDP1 684/4885ALDH1A1 146/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.