SCHEMBL15313667

SCHEMBL15313667

COc1c(Br)cc(C2OCCO2)c(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 5/20 0.42
CA4 P22748 5/20 0.42
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CA1 P00915 4/20 0.33
CA6 P23280 4/20 0.33
HTR2A P28223 4/20 0.33
TTR P02766 1/20 0.32
INSR P06213 1/20 0.32
IGF1R P08069 1/20 0.32
HTR2C P28335 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PTPN1 P18031 2/20 0.31
TPMT P51580 1/20 0.31
ACHE P22303 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15313665 0.76 LMNA (0.36) CA2NPC1RAB9ACA1SMN1; SMN2
SCHEMBL6737359 0.76 ACHE (0.40) NPC1RAB9APTPN1ACHEMAPT
SCHEMBL6040717 0.75 HTR2C (0.47) NPC1RAB9AHTR2AHTR2CALDH1A1
SCHEMBL20263723 0.74 NPC1 (0.32) NPC1RAB9A
SCHEMBL29654713 0.73 HTR2C (0.45) NPC1RAB9AHTR2AHTR2CTP53
SCHEMBL515378 0.73 HTR2C (0.45) NPC1RAB9AHTR2AHTR2CTP53
SCHEMBL6070144 0.72 EGFR (0.40) SMN1; SMN2PTPN1ACHEALDH1A1
SCHEMBL18198243 0.71 NPC1 (0.54) CA2NPC1RAB9ACA1HTR2C
SCHEMBL6711039 0.71 HTR2C (0.56) NPC1RAB9AHTR2AHTR2C
SCHEMBL25384659 0.71 TUBB4A (0.35) CA2CA4NPC1RAB9ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed