SCHEMBL15344337

SCHEMBL15344337

NCc1ccc(CNC(=O)Nc2ccc(CNC(=O)c3ccc(C(=O)NCc4ccc(NC(=O)NCc5ccc(CN)cc5)cc4)cc3)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.63
HDAC6 Q9UBN7 2/20 0.63
NPC1 O15118 1/20 0.58
NAMPT P43490 14/20 0.56
ROCK2 O75116 1/20 0.56
ALDH1A1 P00352 1/20 0.56
EPHX2 P34913 1/20 0.55
NR1H4 Q96RI1 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16383046 0.93 NPC1 (0.71) HDAC1HDAC6NPC1NAMPTALDH1A1
SCHEMBL7119894 0.87 HDAC6 (0.66) HDAC1HDAC6EPHX2NR1H4
SCHEMBL15344288 0.87 HDAC1 (0.58) HDAC1HDAC6NPC1NAMPTALDH1A1
SCHEMBL4743832 0.84 CA2 (0.67) NPC1NAMPTROCK2
SCHEMBL23747520 0.83 RAB9A (0.73) NPC1NAMPTEPHX2
SCHEMBL16378812 0.83 NPC1 (0.64) HDAC1HDAC6NPC1ROCK2ALDH1A1
SCHEMBL26546719 0.83 RAB9A (0.73) NPC1NAMPTALDH1A1
SCHEMBL15344287 0.83 NAMPT (0.56) HDAC1HDAC6NPC1NAMPTALDH1A1
SCHEMBL15344336 0.82 NAMPT (0.55) HDAC1HDAC6NPC1NAMPTEPHX2
Hydrochloric Acid SCHEMBL23728048 0.82 RAB9A (0.71) NPC1NAMPTEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9084735-B2 Self-assembling bis-urea compounds for drug delivery INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2015-07-21 US disclosed
US-20150037390-A1 SELF-ASSEMBLING BIS-UREA COMPOUNDS FOR DRUG DELIVERY AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-02-05 US disclosed
US-8921426-B2 Cationic bis-urea compounds as effective antimicrobial agents INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-12-30 US disclosed
US-20130281515-A1 CATIONIC BIS-UREA COMPOUNDS AS EFFECTIVE ANTIMICROBIAL AGENTS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2013-10-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130281515-A1 CATIONIC BIS-UREA COMPOUNDS AS EFFECTIVE ANTIMICROBIAL AGENTS NOS3, NOS1, NOS2 HDAC1 965/4885HDAC6 685/4885NPC1 1499/4885
US-20150037390-A1 SELF-ASSEMBLING BIS-UREA COMPOUNDS FOR DRUG DELIVERY SLC14A1, NONO, PUF60 HDAC1 550/4885HDAC6 503/4885NPC1 1467/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.