SCHEMBL154274

SCHEMBL154274

NC(CCn1c(=O)cc[nH]c1=O)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.47
GRM2 Q14416 1/20 0.47
GRM8 O00222 1/20 0.41
GRM4 Q14833 1/20 0.41
GRIA1 P42261 4/20 0.40
GRIK1 P39086 2/20 0.40
GRIA2 P42262 3/20 0.39
GRIA3 P42263 3/20 0.39
GRIA4 P48058 3/20 0.39
TYR P14679 2/20 0.38
GRIK2 Q13002 1/20 0.38
GRIK3 Q13003 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28838403 0.86 GRM5 (0.37) GRM5GRM2GRM8GRM4GRIA1
SCHEMBL5282402 0.84 GRIA1 (0.51) GRM5GRIA1GRIK1GRIA2GRIA3
SCHEMBL9694567 0.81 ALDH1A1 (0.33)
SCHEMBL4348692 0.77 ADRA1D (0.37)
D-Glutamate SCHEMBL28865803 0.75 GRM8 (0.51) GRM5GRM2GRM8GRM4GRIA1
SCHEMBL2983409 0.74 ADRA1D (0.34)
SCHEMBL2930015 0.74 HASPIN (0.35)
SCHEMBL17371774 0.74 FABP4 (0.50)
SCHEMBL337058 0.73 TYMP (0.37)
SCHEMBL2899641 0.73 APEX1 (0.48) GRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2056 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9725474-B2 Modified nucleic acid TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-08 US claimed
US-20170175129-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS INC (US) 2017-06-22 US claimed
US-20170136131-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF Modema Therapeutics, Inc. (US) 2017-05-18 US claimed
EP-3157572-A2 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF Moderna Therapeutics, Inc. (US) 2017-04-26 EP claimed
CN-106170553-A Modified nucleic acid molecules and uses thereof 现代治疗公司 2016-11-30 CN claimed
US-20160304552-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. 2016-10-20 US claimed
EP-3080289-A2 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF Moderna Therapeutics, Inc. (US) 2016-10-19 EP claimed
WO-2016043661-A1 MODIFIED PEPTIDE NUCLEIC ACIDS AND THEIR USE NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2016-03-24 WO claimed
WO-2015196130-A2 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. (US) 2015-12-23 WO claimed
US-20150307542-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNATX, INC. 2015-10-29 US claimed
EP-2931319-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF Moderna Therapeutics, Inc. (US) 2015-10-21 EP claimed
WO-2015089511-A2 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. (US) 2015-06-18 WO claimed
WO-2014093924-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. (US) 2014-06-19 WO claimed
WO-2013071079-A1 LIN28/LET-7 CRYSTAL STRUCTURES, PURIFICATION PROTOCOLS, AND MOLECULAR PROBES SUITABLE FOR SCREENING ASSAYS AND THERAPEUTICS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-05-16 WO claimed
EP-4748381-A2 PRODUCTS AND COMPOSITIONS Silence Therapeutics GmbH (DE) 2026-05-27 EP disclosed
EP-4748382-A2 PRODUCTS AND COMPOSITIONS Silence Therapeutics GmbH (DE) 2026-05-27 EP disclosed
CN-122095091-A DsRNA for inhibiting LPA gene expression and application thereof 2026-05-26 CN disclosed
WO-2004064737-A2 THERAPEUTICS COMPOSITIONS ALNYLAM PHARMACEUTICALS (US) 2004-08-05 WO disclosed
US-20020137135-A1 Novel NPG-1 gene that is differentially expressed in prostate tumors BETH ISRAEL DEACONESS MEDICAL CENTER, INC., A MASSACHUSETTS CORPORATION 2002-09-26 US disclosed
US-6287777-B1 SEVERAL GENES EXPRESSED DIFFERENTIALLY BETWEEN THE HUMAN PROSTATE CARCINOMA CELL LINES LNCAP AND PC-3, WHICH ARE ANDROGEN-DEPENDENT AND ANDROGEN-INDEPENDENT, RESPECTIVELY, HAVE NOW BEEN ISOLATED. ONE OF THESE GENES, DESIGNATED NPG-1. BETH ISRAEL DEACONESS MEDICAL CENTER 2001-09-11 US disclosed