SCHEMBL15535562

SCHEMBL15535562

Nc1cc(C2CCN(C(=O)O)CC2)ccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.42
GABRD O14764 2/20 0.42
GABRA1 P14867 2/20 0.42
GABRB1 P18505 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA5 P31644 2/20 0.42
GABRA3 P34903 2/20 0.42
GABRA2 P47869 2/20 0.42
GABRB2 P47870 2/20 0.42
GABRA4 P48169 2/20 0.42
GABRE P78334 2/20 0.42
GABRA6 Q16445 2/20 0.42
GABRG1 Q8N1C3 2/20 0.42
GABRG3 Q99928 2/20 0.42
GABRQ Q9UN88 2/20 0.42
TLR9 Q9NR96 1/20 0.42
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
QDPR P09417 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15602663 0.87 QDPR (0.57) TLR9TLR8TLR7QDPRLMNA
SCHEMBL23089242 0.85 GABRP (0.45) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL15534859 0.82 PROKR1 (0.47) QDPRLMNASCD5HDAC3HDAC4
SCHEMBL23212044 0.82 HDAC4 (0.53) TLR9TLR8TLR7QDPRLMNA
SCHEMBL14239680 0.80 GPR119 (0.50)
SCHEMBL29940481 0.79 NOS3 (0.45) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL3178410 0.79 NOS3 (0.45) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1856770 0.78 LMNA (0.55) LMNASCD5SCDHRH3
SCHEMBL14859120 0.78 ESR2 (0.44) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL30783142 0.78 TRPC6 (0.52) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2852584-A1 SUBSTITUTED DIPYRIDYLAMINES AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2015-04-01 EP disclosed
WO-2013174780-A1 SUBSTITUTED DIPYRIDYLAMINES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2013-11-28 WO disclosed