SCHEMBL155509

SCHEMBL155509

NC(=O)CCCCCCC(=O)N(O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.44
KDM4A O75164 2/20 0.43
KDM4C Q9H3R0 2/20 0.43
KDM5A P29375 1/20 0.43
PHF8 Q9UPP1 1/20 0.43
KDM2A Q9Y2K7 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.41
MAPT P10636 3/20 0.41
LMNA P02545 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
GAA P10253 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TP53 P04637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20767991 0.86 ALDH1A1 (0.40) ALOX5KDM4AKDM4CKDM5APHF8
SCHEMBL7196384 0.84 NPC1 (0.53) ALOX5MAPTLMNANPC1ALDH1A1
SCHEMBL10596450 0.84 NPSR1 (0.53) ALOX5KDM4AKDM4CKDM5APHF8
SCHEMBL1769746 0.84 NPSR1 (0.53) ALOX5KDM4AKDM4CKDM5APHF8
SCHEMBL7985994 0.82 ALDH1A1 (0.48) ALOX5LMNANPC1ALDH1A1POLB
SCHEMBL4138868 0.81 NPSR1 (0.55) ALOX5L3MBTL1MAPTLMNATDP1
SCHEMBL20591107 0.81 TBXAS1 (0.45) MAPTLMNAPOLBHDAC3HDAC4
SCHEMBL836988 0.80 TP53 (0.51) ALOX5NPC1ALDH1A1RAB9ATP53
SCHEMBL9834690 0.79 ALOX5 (0.65) ALOX5KDM4AKDM4CKDM5APHF8
SCHEMBL326865 0.76 RAB9A (0.45) ALOX5L3MBTL1NPC1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 80 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015157500-A1 CLASS IIA HDAC INHIBITORS FOR THE TREATMENT OF INFECTION RESEARCH DEVELOPMENT FOUNDATION (US) 2015-10-15 WO claimed
CN-101115495-B Method to enhance the bone formation activity of bmp by RUNX2 acetylation BIORUNX 2011-06-22 CN claimed
US-20250326771-A1 PIPERAZINE DERIVATIVES USEFUL IN HIV THERAPY VIIV HEALTHCARE CO (US) 2025-10-23 US disclosed
US-20240325398-A1 COMBINATION THERAPIES INFINITY PHARMACEUTICALS, INC. 2024-10-03 US disclosed
US-12053482-B2 Oral formulations of cytidine analogs and methods of use thereof CELGENE CORPORATION (US) 2024-08-06 US disclosed
US-11730736-B2 Anticancer agents RAPT THERAPEUTICS, INC. (US) 2023-08-22 US disclosed
US-20230255996-A1 ORAL FORMULATIONS OF CYTIDINE ANALOGS AND METHODS OF USE THEREOF CELGENE CORPORATION 2023-08-17 US disclosed
US-20230241086-A1 ORAL FORMULATIONS OF CYTIDINE ANALOGS AND METHODS OF USE THEREOF CELGENE CORPORATION 2023-08-03 US disclosed
WO-2023017179-A1 METHYLENE QUINUCLIDINONE COMPANION DIAGNOSTICS Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2023-02-16 WO disclosed
US-11571436-B2 Oral formulations of cytidine analogs and methods of use thereof CELGENE CORPORATION (US) 2023-02-07 US disclosed
US-11554123-B2 Compositions and methods for reactivating latent HIV-1 infections SAINT JOSEPH'S UNIVERSITY (US) 2023-01-17 US disclosed
US-20100184812-A1 MUTUAL PRODRUGS AND METHODS TO TREAT CANCER UNIVERSITY OF MARYLAND, BALTIMORE (US) 2010-07-22 US disclosed
EP-2167090-A2 HDAC INHIBITORS AND HORMONE TARGETED DRUGS FOR THE TREATMENT OF CANCER University of Maryland, Baltimore (US) 2010-03-31 EP disclosed
US-20090286752-A1 ORAL FORMULATIONS OF CYTIDINE ANALOGS AND METHODS OF USE THEREOF CELGENE CORPORATION 2009-11-19 US disclosed
WO-2009126662-A1 ADMINISTRATION OF AN INHIBITOR OF HDAC, AN INHIBITOR OF HER-2, AND A SELECTIVE ESTROGEN RECEPTOR MODULATOR SYNDAX PHARMACEUTICALS, INC. (US) 2009-10-15 WO disclosed
EP-1692097-B1 TRICYCLIC HYDROXAMATE AND BENZAMIDE DERIVATIVES, COMPOSITIONS AND METHODS EXONHIT THERAPEUTICS SA (FR) 2009-09-02 EP disclosed
WO-2009065926-A2 NEW ANTICANCER COMPOUNDS SULFIDRIS S.R.L. (IT) 2009-05-28 WO disclosed
WO-2009064300-A1 COMBINATIONS OF HDAC INHIBITORS AND CYTOKINES/GROWTH FACTORS THE JOHNS HOPKINS UNIVERSITY (US) 2009-05-22 WO disclosed
EP-2022492-A1 Anti-cancer pharmaceutical composition Pianezza, Maurizio (IT) 2009-02-11 EP disclosed
WO-2008154402-A2 HDAC INHIBITORS AND HORMONE TARGETED DRUGS FOR THE TREATMENT OF CANCER UNIVERSITY OF MARYLAND, BALTIMORE (US) 2008-12-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250326771-A1 PIPERAZINE DERIVATIVES USEFUL IN HIV THERAPY CCR5, THPO, IL5 ALOX5 1735/4885KDM4A 2433/4885KDM4C 1838/4885
US-12053482-B2 Oral formulations of cytidine analogs and methods of use thereof DCTD, CDA, NT5C2 ALOX5 725/4885KDM4A 3061/4885KDM4C 1789/4885
US-20230241086-A1 ORAL FORMULATIONS OF CYTIDINE ANALOGS AND METHODS OF USE THEREOF DCTD, CDA, NT5C2 ALOX5 725/4885KDM4A 3061/4885KDM4C 1789/4885
US-20090286752-A1 ORAL FORMULATIONS OF CYTIDINE ANALOGS AND METHODS OF USE THEREOF DCTD, CDA, NT5C2 ALOX5 725/4885KDM4A 3061/4885KDM4C 1789/4885
US-20230255996-A1 ORAL FORMULATIONS OF CYTIDINE ANALOGS AND METHODS OF USE THEREOF DCTD, CDA, NT5C2 ALOX5 725/4885KDM4A 3061/4885KDM4C 1789/4885
US-11571436-B2 Oral formulations of cytidine analogs and methods of use thereof DCTD, CDA, NT5C2 ALOX5 725/4885KDM4A 3061/4885KDM4C 1789/4885
US-20100184812-A1 MUTUAL PRODRUGS AND METHODS TO TREAT CANCER RARA, RARB, RARG ALOX5 1186/4885KDM4A 74/4885KDM4C 165/4885
US-20240325398-A1 COMBINATION THERAPIES HDAC1, HDAC4, HDAC2 ALOX5 3730/4885KDM4A 334/4885KDM4C 492/4885
US-11730736-B2 Anticancer agents CCR4, CCR3, CCR1 ALOX5 4026/4885KDM4A 1609/4885KDM4C 2158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.