5,7-Dimethoxyisoflavone

5,7-Dimethoxyisoflavone

SCHEMBL1675985

COc1cc(OC)c2c(=O)c(-c3ccccc3)coc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 1.00
KDM4E B2RXH2 6/20 1.00
CYP3A4 P08684 5/20 1.00
SMN1; SMN2 Q16637 5/20 1.00
HSD17B10 Q99714 3/20 1.00
MAPT P10636 3/20 1.00
TP53 P04637 3/20 1.00
HPGD P15428 2/20 1.00
THRB P10828 1/20 1.00
NPC1 O15118 4/20 0.82
RAB9A P51151 4/20 0.82
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
NFKB1 P19838 1/20 0.61
CYP2C19 P33261 1/20 0.61
NFKB2 Q00653 1/20 0.61
RELA Q04206 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biochanin A, Dimethyl Ether SCHEMBL5795557 0.90 CYP3A4 (1.00) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL28788159 0.87 KDM4E (0.83) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL31186354 0.86 SMN1; SMN2 (0.76) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL1227819 0.86 SMN1; SMN2 (0.76) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL10622209 0.86 EGFR (0.77) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL30288208 0.85 CYP3A4 (0.81) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
5-Hydroxy-7-Methoxyisoflavone SCHEMBL6142401 0.85 RAB9A (0.83) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL7056427 0.85 CYP3A4 (0.76) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL16335646 0.82 ALDH1A1 (0.69) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10
SCHEMBL16335377 0.82 ALDH1A1 (0.69) ALDH1A1KDM4ECYP3A4SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130245070-A1 COMPOUNDS FOR ENHANCING ARGINASE ACTIVITY AND METHODS OF USING SAME THE RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2013-09-19 US claimed
US-20090253782-A1 Compounds for Enhancing Arginase Activity and Methods of USe Thereof CORNELL RESEARCH FOUNDATION, INC. 2009-10-08 US claimed
WO-2008011083-A2 COMPOUNDS FOR ENHANCING ARGINASE ACTIVITY AND METHODS OF USE THEREOF CORNELL RESEARCH FOUNDATION, INC. (US) 2008-01-24 WO claimed
EP-3013331-B1 MULTITARGET HEDGEHOG PATHWAY INHIBITORS AND THEIR USE FOR THE TREATMENT OF CERTAIN HEDGEHOG (HH)-DEPENDENT TUMORS UNIV DEGLI STUDI DI SIENA (IT) 2023-03-01 EP disclosed
US-20220291237-A1 Gene Expression Inflammatory Age and Its Uses Edifice Health, Inc. (US) 2022-09-15 US disclosed
US-20210030714-A1 COMPOUNDS FOR USE IN THE TREATMENT OF BRAIN DISEASES UNIVERSITA DEGLI STUDI DI ROMA "LA SAPIENZA" (IT) 2021-02-04 US disclosed
EP-3749300-A1 COMPOUNDS FOR USE IN THE TREATMENT OF BRAIN DISEASES Università degli Studi di Roma "La Sapienza" (IT) 2020-12-16 EP disclosed
CN-112004534-A Compounds for use in the treatment of brain tumors 罗马大学 2020-11-27 CN disclosed
WO-2019149962-A1 COMPOUNDS FOR USE IN THE TREATMENT OF BRAIN DISEASES UNIVERSITÀ DEGLI STUDI DI ROMA "LA SAPIENZA" (IT) 2019-08-08 WO disclosed
US-10093642-B2 Multitarget hedgehog pathway inhibitors and uses thereof Università degli Studi di Roma “La Sapienza” (IT) 2018-10-09 US disclosed
US-20160368886-A1 MULTITARGET HEDGEHOG PATHWAY INHIBITORS AND USES THEREOF UNIVERSITA' DEGLI STUDI DI SIENA (IT) 2016-12-22 US disclosed
US-20140186277-A1 Methods and Compositions for Reducing Skin Damage SHISEIDO CO., LTD. (JP) 2014-07-03 US disclosed
US-20130245070-A1 COMPOUNDS FOR ENHANCING ARGINASE ACTIVITY AND METHODS OF USING SAME THE RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2013-09-19 US disclosed
US-20110091387-A1 METHODS AND COMPOSITIONS FOR REDUCING SKIN DAMAGE THE GENERAL HOSPITAL CORPORATION (US) 2011-04-21 US disclosed
CN-101918037-A Be used to reduce the method and composition of skin injury GEN HOSPITAL CORP 2010-12-15 CN disclosed
US-20090269772-A1 SYSTEMS AND METHODS FOR IDENTIFYING COMBINATIONS OF COMPOUNDS OF THERAPEUTIC INTEREST THERASIS, INC. 2009-10-29 US disclosed
US-20090253782-A1 Compounds for Enhancing Arginase Activity and Methods of USe Thereof CORNELL RESEARCH FOUNDATION, INC. 2009-10-08 US disclosed
US-20090143279-A1 Methods and compositions for treating metabolic disorders PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2009-06-04 US disclosed
WO-2009065141-A1 METHODS AND COMPOSITIONS FOR REDUCING SKIN DAMAGE THE GENERAL HOSPITAL CORPORATION (US) 2009-05-22 WO disclosed
WO-2008011083-A2 COMPOUNDS FOR ENHANCING ARGINASE ACTIVITY AND METHODS OF USE THEREOF CORNELL RESEARCH FOUNDATION, INC. (US) 2008-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160368886-A1 MULTITARGET HEDGEHOG PATHWAY INHIBITORS AND USES THEREOF SHH, GLI1, SMO ALDH1A1 2823/4885KDM4E 942/4885CYP3A4 4845/4885
US-20130245070-A1 COMPOUNDS FOR ENHANCING ARGINASE ACTIVITY AND METHODS OF USING SAME ARG2, ARG1, OTC ALDH1A1 249/4885KDM4E 1426/4885CYP3A4 3922/4885
US-10093642-B2 Multitarget hedgehog pathway inhibitors and uses thereof SHH, GLI1, SMO ALDH1A1 2823/4885KDM4E 942/4885CYP3A4 4845/4885
US-20210030714-A1 COMPOUNDS FOR USE IN THE TREATMENT OF BRAIN DISEASES NLN, ADCYAP1R1, PYGB ALDH1A1 1323/4885KDM4E 2941/4885CYP3A4 3645/4885
US-20090143279-A1 Methods and compositions for treating metabolic disorders PC, PCK2, CS ALDH1A1 860/4885KDM4E 3739/4885CYP3A4 2876/4885
US-20090253782-A1 Compounds for Enhancing Arginase Activity and Methods of USe Thereof ARG2, ARG1, OTC ALDH1A1 292/4885KDM4E 1521/4885CYP3A4 3582/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.