SCHEMBL16795137

SCHEMBL16795137

CN1CCC(NCc2cc(O)cc(B3OC(C)(C)C(C)(C)O3)c2)CC1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.34
BACE1 P56817 5/20 0.34
PDGFRB P09619 1/20 0.34
KDR P35968 1/20 0.34
MAP4K4 O95819 2/20 0.33
CARM1 Q86X55 5/20 0.33
PRMT6 Q96LA8 5/20 0.33
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD5 P21918 1/20 0.32
BCHE P06276 3/20 0.32
PRMT8 Q9NR22 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
CHEK1 O14757 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16795329 0.88 ALDH1A1 (0.43) ALDH1A1TSHRCYP2D6
SCHEMBL16795221 0.86 HRH3 (0.40) ACHEBACE1CARM1PRMT6BCHE
SCHEMBL18580408 0.82 LPL (0.47) ACHEBACE1MAP4K4CARM1PRMT6
SCHEMBL18580127 0.82 LPL (0.46) ACHEBACE1CARM1PRMT6BCHE
SCHEMBL16795407 0.78 KDM4E (0.44) MAP4K4ALDH1A1TSHR
SCHEMBL16795229 0.75 CXCR3 (0.36) ACHEBACE1BCHEALDH1A1
SCHEMBL16795291 0.75 CARM1 (0.47) ACHEBACE1PDGFRBKDRMAP4K4
SCHEMBL16795129 0.70 MAOB (0.36) DRD2ALDH1A1
SCHEMBL18579622 0.69 LIPG (0.48) ACHEBACE1MAP4K4CARM1PRMT6
SCHEMBL18579621 0.69 LIPG (0.48) ACHEBACE1MAP4K4CARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015086693-A1 PYRAZOLOPYRIMIDIN-2-YL DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2015-06-18 WO disclosed