SCHEMBL16795407

SCHEMBL16795407

CN1CCC(N(C)Cc2cc(O)cc(B3OC(C)(C)C(C)(C)O3)c2)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
NOS2 P35228 6/20 0.38
NOS3 P29474 5/20 0.38
NOS1 P29475 5/20 0.38
LTA4H P09960 1/20 0.38
MAP4K4 O95819 2/20 0.34
TSHR P16473 1/20 0.33
AKT1 P31749 1/20 0.31
LPL P06858 1/20 0.30
LIPG Q9Y5X9 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16795137 0.78 ACHE (0.34) ALDH1A1MAP4K4TSHR
SCHEMBL16795390 0.75 NOS2 (0.53) KDM4EALDH1A1NOS2NOS3NOS1
SCHEMBL18953910 0.71 LPL (0.51) LTA4HLPLLIPG
SCHEMBL16795129 0.69 MAOB (0.36) KDM4EALDH1A1KMT2A
SCHEMBL16795410 0.68 L3MBTL3 (0.42) KDM4EALDH1A1TSHRKMT2A
SCHEMBL14680428 0.68 ALDH1A1 (0.55) KDM4EALDH1A1NOS2NOS3NOS1
SCHEMBL16795329 0.68 ALDH1A1 (0.43) KDM4EALDH1A1TSHRLPLLIPG
SCHEMBL16426120 0.68 LPL (0.44) LPLLIPG
SCHEMBL28628663 0.68 LPL (0.44) LPLLIPG
SCHEMBL16795229 0.67 CXCR3 (0.36) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015086693-A1 PYRAZOLOPYRIMIDIN-2-YL DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2015-06-18 WO disclosed