SCHEMBL1702773

SCHEMBL1702773

N#Cc1c(Cl)ccnc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.42
CYP3A4 P08684 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
BCL6 P41182 3/20 0.38
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 4/20 0.38
LMNA P02545 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
KMO O15229 1/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
MAPK1 P28482 3/20 0.36
KMT2A Q03164 5/20 0.35
HPGD P15428 3/20 0.35
MAPT P10636 3/20 0.35
MEN1 O00255 3/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30072681 1.00 LRRK2 (0.42) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL20568819 0.79 BCL6 (0.34) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL15741185 0.78 LRRK2 (0.40) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL20836128 0.78 CYP11B2 (0.41) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL2937411 0.78 LRRK2 (0.40) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL1698600 0.78 NTRK1 (0.42) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL15741203 0.78 LRRK2 (0.40) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL31622333 0.78 LRRK2 (0.40) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL5802874 0.78 KCNMA1 (0.40) LRRK2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL677194 0.78 L3MBTL1 (0.45) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 186 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4741392-A1 1H-PYRAZOLO[4,3-C]PYRIDINE COMPOUND, AND COMPOSITION THEREOF AND USE THEREOF Shenzhen TargetRx Co., Ltd. (CN) 2026-05-13 EP disclosed
EP-4729127-A2 BCL6 INHIBITORS Cancer Research Technology Limited (GB) 2026-04-22 EP disclosed
US-20260042776-A1 BCL6 INHIBITORS CANCER RESEARCH TECH LTD (GB) 2026-02-12 US disclosed
US-12528816-B2 Substituted imidazo [1,2-b] pyridazines and [1, 2, 4] triazolo [ 4,3-b] pyridazines as camkii inhibitors CARDURION PHARMACEUTICALS, INC. (US) 2026-01-20 US disclosed
US-12486285-B2 BCL6 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2025-12-02 US disclosed
US-20250163076-A1 SYNTHESIS OF BRUTON'S TYROSINE KINASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2025-05-22 US disclosed
US-20250127906-A1 SMALL-MOLECULE DEGRADERS OF CDK8 AND CDK19 UNIVERSITY OF SOUTH CAROLINA 2025-04-24 US disclosed
US-20250115598-A1 BIFUNCTIONAL ARYLSULPHONAMIDE COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2025-04-10 US disclosed
US-20250059188-A1 ARYLSULPHONAMIDE COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2025-02-20 US disclosed
WO-2025007863-A1 1H-PYRAZOLO[4,3-C]PYRIDINE COMPOUND, AND COMPOSITION THEREOF AND USE THEREOF 深圳市塔吉瑞生物医药有限公司 2025-01-09 WO disclosed
US-6197964-B1 CHLORINATION USING BASIC CATALYST; DESALTING, HYDROLYSIS BAYER AKTIENGESELLSCHAFT (DE) 2001-03-06 US disclosed
US-6046207-A FOR INHIBITING ALPHA-1 ADRENORECEPTORS AND TREATING BENIGN PROSTATIC HYPERPLASIA, ALSO CALLED BENIGN PROSTATIC HYPERTROPHY, OR OTHER UROLOGICAL OR GYNECOLOGICAL DISEASES SUCH AS BLADDER OUTLET OBSTRUCTION, NEUROGENIC BLADDER ABBOTT LABORATORIES 2000-04-04 US disclosed
WO-1999062908-A2 CELL ADHESION-INHIBITING ANTINFLAMMATORY COMPOUNDS ABBOTT LABORATORIES (US) 1999-12-09 WO disclosed
EP-0942911-A1 BENZOPYRANOPYRROLE AND BENZOPYRANOPYRIDINE ALPHA-1 ADRENERGIC COMPOUNDS Abbott Laboratories (US) 1999-09-22 EP disclosed
US-5891882-A TREATING BENIGN PROSTATIC HYPERPLASIA OR OTHER UROLOGICAL DISEASES SUCH AS BLADDER OUTLET OBSTRUCTION AND NEUROGENIC BLADDER, OR GYNECOLOGICAL SYNDROMES SUCH AS DYSMENORRHEA ABBOTT LABORATORIES (US) 1999-04-06 US disclosed
WO-1998024791-A1 BENZOPYRANOPYRROLE AND BENZOPYRANOPYRIDINE ALPHA-1 ADRENERGIC COMPOUNDS ABBOTT LABORATORIES (US) 1998-06-11 WO disclosed
US-5710157-A INSECTICIDES FOR AGRICULTURE FMC CORPORATION (US) 1998-01-20 US disclosed
US-5593998-A 2,4-diamino-5,6-disubstituted-and 5,6,7-trisubstituted-5-deazapteridines as insecticides FMC CORPORATION (US) 1997-01-14 US disclosed
US-5547954-A MIXED WITH AGRICULTURAL ACCEPTABLE CARRIER FMC CORPORATION (US) 1996-08-20 US disclosed
US-5532370-A FOR INSECTS INCLUDING LARVAE SUCH AS TOBACCO BUDWORM FMC CORPORATION (US) 1996-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12528816-B2 Substituted imidazo [1,2-b] pyridazines and [1, 2, 4] triazolo [ 4,3-b] pyridazines as camkii inhibitors RYR2, CACNA1C, CAMK4 LRRK2 1697/4885CYP3A4 2634/4885CYP1A2 1551/4885
US-20250127906-A1 SMALL-MOLECULE DEGRADERS OF CDK8 AND CDK19 CDK8, CDK9, CDK18 LRRK2 980/4885CYP3A4 3460/4885CYP1A2 4043/4885
US-20250163076-A1 SYNTHESIS OF BRUTON'S TYROSINE KINASE INHIBITORS ABL1, BTK, LYN LRRK2 291/4885CYP3A4 3534/4885CYP1A2 2799/4885
US-20250115598-A1 BIFUNCTIONAL ARYLSULPHONAMIDE COMPOUNDS MLKL, CASP1, CASP9 LRRK2 21/4885CYP3A4 1314/4885CYP1A2 1645/4885
US-12486285-B2 BCL6 inhibitors BCL6, BCL6B, BCL3 LRRK2 1478/4885CYP3A4 3422/4885CYP1A2 3289/4885
US-20260042776-A1 BCL6 INHIBITORS BCL6, BCL6B, BCL9 LRRK2 1049/4885CYP3A4 3867/4885CYP1A2 3720/4885
US-20250059188-A1 ARYLSULPHONAMIDE COMPOUNDS MLKL, CASP1, CASP9 LRRK2 31/4885CYP3A4 1822/4885CYP1A2 2336/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.