SCHEMBL1704989

SCHEMBL1704989

Cc1cc(Nc2cccc(-c3cccc(C4=CCN(C(=O)OC(C)(C)C)CC4)c3)n2)nn1C(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.44
JAK1 P23458 1/20 0.43
GRM1 Q13255 10/20 0.43
GRM5 P41594 9/20 0.43
PDK4 Q16654 1/20 0.42
SOS1 Q07889 1/20 0.42
CDK7 P50613 1/20 0.41
CDK13 Q14004 1/20 0.41
CDK12 Q9NYV4 1/20 0.41
LIPC P11150 1/20 0.40
LIPG Q9Y5X9 1/20 0.40
CYP11B2 P19099 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704903 0.91 GRM1 (0.45) NAMPTJAK1GRM1GRM5PDK4
SCHEMBL902774 0.90 ALDH1A1 (0.37) SOS1
SCHEMBL1704197 0.86 KARS1 (0.49) NAMPTJAK1GRM1GRM5
SCHEMBL1704146 0.85 NAMPT (0.43) NAMPTJAK1GRM1GRM5PDK4
SCHEMBL1705279 0.83 GRM1 (0.47) NAMPTJAK1GRM1GRM5PDK4
SCHEMBL1704583 0.82 ADORA2A (0.48)
SCHEMBL1704634 0.81 ALDH1A1 (0.38) NAMPT
SCHEMBL1705277 0.81 JAK2 (0.44) NAMPT
SCHEMBL901325 0.79 GRM1 (0.50) NAMPTJAK1GRM1GRM5PDK4
SCHEMBL7831576 0.76 PDK4 (0.58) NAMPTGRM1GRM5PDK4SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed