SCHEMBL902774

SCHEMBL902774

Cc1cc(Nc2cccc(-c3cccc(C4=CCN(C(=O)O)CC4)c3)n2)nn1C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
QDPR P09417 1/20 0.36
MAPT P10636 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
SOS1 Q07889 1/20 0.35
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
KARS1 Q15046 4/20 0.35
LMNA P02545 2/20 0.35
HTT P42858 2/20 0.35
HPGD P15428 2/20 0.35
USP2 O75604 1/20 0.35
LIMK1 P53667 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704634 0.91 ALDH1A1 (0.38) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL1704989 0.90 NAMPT (0.44) SOS1
SCHEMBL902789 0.84 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL901312 0.83 KARS1 (0.54) ALDH1A1SMN1; SMN2KARS1
SCHEMBL1704903 0.82 GRM1 (0.45) SOS1
SCHEMBL1704829 0.81 KARS1 (0.43) ALDH1A1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL902923 0.79 NPC1 (0.36) ALDH1A1KDM4ENPC1RAB9AKARS1
SCHEMBL1704842 0.79 KARS1 (0.52) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL902090 0.78 KARS1 (0.55) KARS1
SCHEMBL1704197 0.75 KARS1 (0.49) KARS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed