SCHEMBL172474

SCHEMBL172474

CCc1nn2ccc3oc(C)cc3c2c1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.38
HTR2C P28335 4/20 0.38
MTNR1A P48039 2/20 0.33
MTNR1B P49286 2/20 0.33
SLC22A12 Q96S37 1/20 0.32
POLB P06746 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
THRB P10828 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
TBXAS1 P24557 1/20 0.31
PRNP P04156 1/20 0.31
TP53 P04637 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 3/20 0.31
HPGD P15428 2/20 0.31
FABP3 P05413 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL126198 0.87 ALDH1A1 (0.39) HTR2AHTR2CTDP1L3MBTL1MEN1
SCHEMBL124840 0.80 HTR2C (0.39) HTR2AHTR2CMTNR1AMTNR1BTHRB
SCHEMBL124536 0.76 HTR2C (0.40) HTR2AHTR2CMTNR1AMTNR1B
SCHEMBL126955 0.75 HTR2A (0.37) HTR2AHTR2CMTNR1AMTNR1B
SCHEMBL2053937 0.73 POLB (0.37) MTNR1AMTNR1BPOLBTDP1L3MBTL1
SCHEMBL172150 0.68 MTNR1B (0.63) HTR2AMTNR1AMTNR1B
SCHEMBL13851431 0.68 ALOX15 (0.36) MTNR1AMTNR1BPOLBTDP1L3MBTL1
SCHEMBL19514014 0.66 FABP4 (0.42) SLC22A12MEN1KMT2AKDM4EFABP3
SCHEMBL28437880 0.66 GABRP (0.38) MTNR1AMTNR1BSLC22A12POLBTDP1
SCHEMBL21584617 0.66 PTGDR2 (0.37) SLC22A12MEN1KMT2ASMN1; SMN2PRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100895-B1 TRICYCLIC COMPOUND AND MEDICAL USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2012-03-07 EP disclosed
EP-2100895-A1 TRICYCLIC COMPOUND AND MEDICAL USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-09-16 EP disclosed