SCHEMBL1729370

SCHEMBL1729370

CNC(CN(CC=O)C(=O)O)C1CCN(c2ccc3ccc(Cl)cc3n2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.43
PDE10A Q9Y233 2/20 0.41
PDE2A O00408 1/20 0.41
HTR3A P46098 3/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
HRH4 Q9H3N8 2/20 0.36
DGAT1 O75907 2/20 0.35
KCNH2 Q12809 2/20 0.35
OPRK1 P41145 1/20 0.35
ADORA2A P29274 1/20 0.34
SMO Q99835 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ACACB O00763 1/20 0.33
HSD11B1 P28845 1/20 0.33
P2RX7 Q99572 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1729308 0.95 HRH3 (0.44) HRH3PDE10APDE2AHTR3AHTR3E
SCHEMBL1728165 0.89 KDM4E (0.45) HRH3PDE10APDE2AHTR3AHTR3E
SCHEMBL1730418 0.87 HRH3 (0.45) HRH3PDE10APDE2AHTR3AHTR3E
SCHEMBL1729779 0.87 SMO (0.34) PDE10APDE2ADGAT1KCNH2ADORA2A
SCHEMBL1727892 0.86 HTR1A (0.39) HRH3HTR3ASMOKDM4EALDH1A1
SCHEMBL1728927 0.84 HRH3 (0.47) HRH3KCNH2KDM4EALDH1A1ACACB
SCHEMBL1729592 0.84 PTGES (0.42) PDE10APDE2ASMOHSD11B1PTGES
SCHEMBL1728881 0.83 HCAR2 (0.36) PDE10AOPRK1SMOKDM4EALDH1A1
SCHEMBL1727558 0.83 KCNH2 (0.40) DGAT1KCNH2ADORA2AKDM4E
SCHEMBL1729453 0.82 PDE10A (0.36) PDE10AHTR3AHRH4OPRK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP claimed