SCHEMBL1734492

SCHEMBL1734492

c1ccc(CC[N]C2CCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
SLC18A2 Q05940 1/20 0.44
TRPA1 O75762 1/20 0.42
CYP2E1 P05181 1/20 0.42
CYP2A6 P11509 1/20 0.42
MIF P14174 1/20 0.42
HIF1A Q16665 1/20 0.42
CYP2A13 Q16696 1/20 0.42
EPAS1 Q99814 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2241838 0.75 GRIN1 (0.42) TRPA1MIF
SCHEMBL1796446 0.73 GRIN1 (0.45) TRPA1MIF
SCHEMBL5122547 0.72 LOXL2 (0.43) HIF1AHRH3
SCHEMBL2242592 0.70 ALDH1A1 (0.41) TRPA1MIFHRH3
SCHEMBL7756938 0.68 OPRM1 (0.58) OPRM1OPRD1OPRK1SLC18A2
SCHEMBL4524677 0.68 MIF (0.47) OPRM1OPRD1OPRK1TRPA1CYP2E1
SCHEMBL6335562 0.68 HIF1A (0.56) TRPA1CYP2E1CYP2A6MIFHIF1A
SCHEMBL721250 0.68 HIF1A (0.56) TRPA1CYP2E1CYP2A6MIFHIF1A
Cyclooctane SCHEMBL18187569 0.67 SIGMAR1 (0.58) CYP2A6
SCHEMBL4816295 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8759584-B2 Synthesis of biguanidines and triazines, and biguanidino-aluminium complexes as intermediates BAYER CROPSCIENCE AG (DE) 2014-06-24 US disclosed
EP-2231679-B1 SYNTHESIS OF BIGUANIDINES AND TRIAZINES, AND BIGUANIDINO-ALUMINIUM COMPLEXES AS INTERMEDIATES BAYER CROPSCIENCE AG (DE) 2011-11-16 EP disclosed
US-20100305317-A1 SYNTHESIS OF BIGUANIDINES AND TRIAZINES, AND BIGUANIDINO-ALUMINIUM COMPLEXES AS INTERMEDIATES BAYER CROPSCIENCE AG (DE) 2010-12-02 US disclosed
EP-2070934-A1 Synthesis of biguanidines and triazines, and biguanidino-aluminium complexes as intermediates Bayer CropScience AG (DE) 2009-06-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100305317-A1 SYNTHESIS OF BIGUANIDINES AND TRIAZINES, AND BIGUANIDINO-ALUMINIUM COMPLEXES AS INTERMEDIATES ATIC, SRM, F12 OPRM1 2689/4885OPRD1 3967/4885OPRK1 3859/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.