SCHEMBL1758271

SCHEMBL1758271

CC(C)(C)ONCC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.35
HMGCR P04035 1/20 0.35
CHRM1 P11229 1/20 0.35
TBXA2R P21731 1/20 0.35
ADRA1A P35348 1/20 0.35
CTH P32929 1/20 0.34
CYP2D6 P10635 2/20 0.33
TSHR P16473 2/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
APEX1 P27695 1/20 0.33
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
PTGS2 P35354 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
LDHA P00338 1/20 0.32
SRR Q9GZT4 1/20 0.32
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19901566 0.83 EGLN1 (0.39) EGLN1CTHAPEX1ALDH1A1MAPT
SCHEMBL11923002 0.78 MAOA (0.41)
SCHEMBL13140609 0.76 LMNA (0.38) ALDH1A1MAPTLMNA
SCHEMBL27764506 0.76 ALDH1A1 (0.34) EGLN1SMN1; SMN2CYP2D6ALDH1A1
SCHEMBL31612137 0.75 EGLN1 (0.33) EGLN1SMN1; SMN2CTHTSHRLDHA
Oxalic Acid SCHEMBL1052746 0.73 POLB (0.34) ALDH1A1KDM4E
SCHEMBL9059109 0.73 DGAT1 (0.34) EGLN1HMGCRCHRM1TBXA2RADRA1A
SCHEMBL13118699 0.72 MEN1 (0.37) ADRA1ATSHRALDH1A1LMNATDP1
SCHEMBL17177603 0.72 NOS2 (0.32)
SCHEMBL1287256 0.71 EGLN1 (0.35) EGLN1SMN1; SMN2HMGCRCHRM1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119684406-A Enzyme response self-assembled polypeptide prodrug loaded with camptothecine, preparation and application thereof 东南大学 2025-03-25 CN disclosed
WO-2023150540-A1 HYDROXAMIC ACID MACROCYCLIC AGENTS WITH PENDANT CHELATING MOIETIES AND COMPLEXES THEREOF LUMIPHORE, INC. (US) 2023-08-10 WO disclosed
CN-104650342-B Highly branched chain polymeric drug precursor and its application 江苏豪森药业集团有限公司 2018-07-10 CN disclosed
US-9650664-B2 Use of photocleavable compounds FEMTONICS KFT (HU) 2017-05-16 US disclosed
CN-104650342-A Highly-branched polymerized prodrug, and applications thereof JIANGSU HANSOH PHARMACEUTICAL 2015-05-27 CN disclosed
US-20140234883-A1 USE OF PHOTOCLEAVABLE COMPOUNDS FEMTONICS KFT (HU) 2014-08-21 US disclosed
EP-2763965-A2 USE OF PHOTOCLEAVABLE COMPOUNDS Femtonics Kft. (HU) 2014-08-13 EP disclosed
WO-2013050798-A2 USE OF PHOTOCLEAVABLE COMPOUNDS FEMTONICS KFT. (HU) 2013-04-11 WO disclosed
EP-1758916-B1 3-BETA-D-RIBOFURANOSYLTHIAZOLO[4,5-d]PYRIDIMINE NUCLEOSIDES AND USES THEREOF ANADYS PHARMACEUTICALS INC (US) 2012-11-21 EP disclosed
EP-1512683-B1 Novel opiate compounds, methods of making and methods of use RES TRIANGLE INST (US) 2011-08-31 EP disclosed
US-20020193602-A1 Novel opiate compounds, methods of making and methods of use RESEARCH TRIANGLE INSTITUTE (US) 2002-12-19 US disclosed
US-20020169324-A1 NOVEL OPIATE COMPOUNDS, METHODS OF MAKING AND METHODS OF USE RESEARCH TRIANGLE INSTITUTE (US) 2002-11-14 US disclosed
US-20020165396-A1 NOVEL OPIATE COMPOUNDS, METHODS OF MAKING AND METHODS OF USE RESEARCH TRIANGLE INSTITUTE (US) 2002-11-07 US disclosed
EP-1061919-A4 NOVEL OPIATE COMPOUNDS, METHODS OF MAKING AND METHODS OF USE RES TRIANGLE INST (US) 2002-09-04 EP disclosed
EP-1061919-A1 NOVEL OPIATE COMPOUNDS, METHODS OF MAKING AND METHODS OF USE Carrol, Frank Ivy (US) 2000-12-27 EP disclosed
US-5990278-A REACTING AN ORGANIC CARBOXYLIC ACID WITH AN AMINE DERIVATIVE CONTAINING A PROTECTIVE GROUP TO FORM PROTECTED CARBAMIDE, REACTING PROTECTED CARBAMIDE AT A FIRST PH TO SPLIT OFF PROTECTIVE GROUP, REACTING IN SECOND PH TO FORM CARBAMIDE HOFFMANN STEFEN (DE) 1999-11-23 US disclosed
WO-1999045925-A1 NOVEL OPIATE COMPOUNDS, METHODS OF MAKING AND METHODS OF USE RESEARCH TRIANGLE INSTITUTE (US) 1999-09-16 WO disclosed
EP-0506478-A1 Piperidine derivatives ELI LILLY AND COMPANY (US) 1992-09-30 EP disclosed
CN-1048030-A Promote the phenol derivatives of growth factor of human nerve SANKYO CO (JP) 1990-12-26 CN disclosed
EP-0399814-A2 Phenol derivatives for promoting human nerve growth factor Sankyo Company Limited (JP) 1990-11-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020169324-A1 NOVEL OPIATE COMPOUNDS, METHODS OF MAKING AND METHODS OF USE OPRK1, OPRM1, OPRL1 EGLN1 2784/4885SMN1; SMN2 2062/4885HMGCR 2451/4885
US-20020193602-A1 Novel opiate compounds, methods of making and methods of use OPRK1, OPRM1, OPRL1 EGLN1 2784/4885SMN1; SMN2 2062/4885HMGCR 2451/4885
US-20020165396-A1 NOVEL OPIATE COMPOUNDS, METHODS OF MAKING AND METHODS OF USE OPRK1, OPRM1, OPRL1 EGLN1 2784/4885SMN1; SMN2 2062/4885HMGCR 2451/4885
US-20140234883-A1 USE OF PHOTOCLEAVABLE COMPOUNDS ERCC1, ERCC4, ERCC5 EGLN1 1084/4885SMN1; SMN2 4211/4885HMGCR 1361/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.