D-Glutamate

D-Glutamate

SCHEMBL1782280

N[C@@H](CCC(=O)O)C(=O)[O-].N[C@@H](CCC(=O)O)C(=O)[O-].[Na+].[Na+]

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of D-Glutamate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP known ✓ O00591 2/20 0.50
GABRD known ✓ O14764 2/20 0.50
GABRA1 known ✓ P14867 2/20 0.50
GABRB1 known ✓ P18505 2/20 0.50
GABRG2 known ✓ P18507 2/20 0.50
GABRB3 known ✓ P28472 2/20 0.50
GABRA5 known ✓ P31644 2/20 0.50
GABRA3 known ✓ P34903 2/20 0.50
GABRA2 known ✓ P47869 2/20 0.50
GABRB2 known ✓ P47870 2/20 0.50
GABRA4 known ✓ P48169 2/20 0.50
GABRE known ✓ P78334 2/20 0.50
GABRA6 known ✓ Q16445 2/20 0.50
GABRG1 known ✓ Q8N1C3 2/20 0.50
GABRG3 known ✓ Q99928 2/20 0.50
GABRQ known ✓ Q9UN88 2/20 0.50
CYP1A2 P05177 2/20 0.62
GRM8 O00222 1/20 0.62
GRM6 O15303 1/20 0.62
GRIN2D O15399 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
D-Glutamate SCHEMBL27981176 1.00 CYP1A2 (0.62) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL1532402 1.00 CYP1A2 (0.62) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL541430 1.00 CYP1A2 (0.62) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL16336 1.00 CYP1A2 (0.62) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL23828179 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL31067339 0.98 GRM8 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL2853216 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL3781140 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL317907 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL30149979 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8343563-B2 Egg-filled food product CARGILL, INCORPORATED (US) 2013-01-01 US disclosed
US-20110117253-A1 EGG-FILLED FOOD PRODUCT CARGILL, INCORPORATED (US) 2011-05-19 US disclosed
US-20060121160-A1 Egg-filled food product CARGILL, INCORPORATED 2006-06-08 US disclosed
WO-2006060812-A1 EGG-FILLED FOOD PRODUCT CARGILL, INCORPORATED (US) 2006-06-08 WO disclosed