Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | HTR1B | P28222 | 2/20 | 0.39 |
| ▸ | HTR1D | P28221 | 1/20 | 0.39 |
| ▸ | SIGMAR1 | Q99720 | 1/20 | 0.39 |
| ▸ | HTR7 | P34969 | 7/20 | 0.38 |
| ▸ | GPR84 | Q9NQS5 | 1/20 | 0.38 |
| ▸ | MTNR1A | P48039 | 1/20 | 0.38 |
| ▸ | MTNR1B | P49286 | 1/20 | 0.38 |
| ▸ | LMNA | P02545 | 1/20 | 0.38 |
| ▸ | PKM | P14618 | 1/20 | 0.38 |
| ▸ | L3MBTL1 | Q9Y468 | 1/20 | 0.37 |
| ▸ | NPC1 | O15118 | 2/20 | 0.37 |
| ▸ | RAB9A | P51151 | 2/20 | 0.37 |
| ▸ | MAPT | P10636 | 1/20 | 0.36 |
| ▸ | SMN1; SMN2 | Q16637 | 1/20 | 0.36 |
| ▸ | DRD2 | P14416 | 1/20 | 0.36 |
| ▸ | DRD4 | P21917 | 1/20 | 0.36 |
| ▸ | DRD3 | P35462 | 1/20 | 0.36 |
| ▸ | ADRA1D | P25100 | 1/20 | 0.36 |
| ▸ | ADRA1A | P35348 | 1/20 | 0.36 |
| ▸ | ADRA1B | P35368 | 1/20 | 0.36 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL17844247 | 0.81 | HTR1B (0.39) | HTR1BHTR1DGPR84MTNR1AMTNR1B | |
| SCHEMBL5185824 | 0.79 | NPBWR1 (0.43) | LMNAL3MBTL1RAB9AMAPTSMN1; SMN2 | |
| SCHEMBL5197239 | 0.77 | GSK3B (0.43) | LMNANPC1RAB9AMAPTSMN1; SMN2 | |
| SCHEMBL3541635 | 0.75 | MAPT (0.49) | LMNAL3MBTL1MAPTSMN1; SMN2 | |
| SCHEMBL5186747 | 0.74 | PTPN2 (0.37) | HTR1BHTR1DGPR84MTNR1AMTNR1B | |
| SCHEMBL17844223 | 0.74 | DRD2 (0.41) | GPR84LMNAL3MBTL1NPC1RAB9A | |
| SCHEMBL5185609 | 0.74 | ALDH1A1 (0.43) | NPC1RAB9AMAPTSMN1; SMN2 | |
| SCHEMBL17844180 | 0.74 | KDM4E (0.37) | LMNANPC1RAB9AMAPTSMN1; SMN2 | |
| SCHEMBL17844238 | 0.73 | SMN1; SMN2 (0.43) | HTR1BHTR1DHTR7LMNAL3MBTL1 | |
| SCHEMBL17844226 | 0.73 | MAPK1 (0.37) | LMNAMAPTSMN1; SMN2 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| WO-2016100619-A2 | TREATMENT AND DIAGNOSIS OF CANCER | RGENIX, INC. (US) | 2016-06-23 | — | — | WO | disclosed |