SCHEMBL17844160

SCHEMBL17844160

CC(C)(C)n1sc(-c2ccccc2)c(NC2CCN(CCc3ccccc3)CC2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.45
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ACHE P22303 3/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA4 P22748 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA13 Q8N1Q1 1/20 0.43
CA14 Q9ULX7 1/20 0.43
DRD4 P21917 3/20 0.41
DRD2 P14416 1/20 0.41
CCR3 P51677 1/20 0.40
FAAH O00519 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844249 0.90 ACHE (0.50) SIGMAR1ALDH1A1GAAACHEDRD4
SCHEMBL17844171 0.89 MALT1 (0.47) ACHEDRD4DRD2BCHE
SCHEMBL17844164 0.86 KAT2B (0.38) CA12CA2CA9
SCHEMBL17844243 0.78 PRKAA2 (0.43) ACHEBCHE
SCHEMBL3546550 0.75 LMNA (0.42) ALDH1A1MEN1KMT2A
SCHEMBL17844145 0.74 HRH3 (0.38) ALDH1A1MEN1KMT2A
SCHEMBL17844110 0.73 MAOA (0.40) SIGMAR1MEN1KMT2A
SCHEMBL17844162 0.72 HRH3 (0.41) ALDH1A1
SCHEMBL1998987 0.71 NR1H2 (0.48) SIGMAR1ALDH1A1GAAHSD17B10ACHE
SCHEMBL5316660 0.70 METAP1 (0.49) ALDH1A1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100619-A2 TREATMENT AND DIAGNOSIS OF CANCER RGENIX, INC. (US) 2016-06-23 WO disclosed