SCHEMBL17848969

SCHEMBL17848969

CCOC(=O)c1ccn(C)c(=O)c1OCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
HPGD P15428 3/20 0.47
ALDH1A1 P00352 2/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
MAOB P27338 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
HSP90AA1 P07900 1/20 0.46
TSHR P16473 3/20 0.45
MAPT P10636 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
PPIA P62937 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
HTT P42858 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2237686 0.92 ALDH1A1 (0.49) HPGDALDH1A1MEN1KMT2ATSHR
SCHEMBL2240565 0.85 HPGD (0.44) HPGDALDH1A1GAAMEN1KMT2A
SCHEMBL19709882 0.84 MAOB (0.48) HPGDALDH1A1MAOBMEN1KMT2A
SCHEMBL19646278 0.84 ALDH1A1 (0.43) KDM4EHPGDALDH1A1GLAGAA
SCHEMBL16789591 0.83 GLRA1 (0.47) HPGDALDH1A1MEN1KMT2ATSHR
SCHEMBL6865199 0.81 HPGD (0.38) HPGDALDH1A1GAAMEN1KMT2A
SCHEMBL757286 0.80 TSHR (0.46) KDM4EHPGDALDH1A1GLAGAA
SCHEMBL6858810 0.80 LIPG (0.47) KDM4EHPGDALDH1A1GLAGAA
SCHEMBL8333370 0.78 LIPG (0.47) KDM4EHPGDALDH1A1GLAGAA
SCHEMBL28877532 0.78 ALDH1A1 (0.56) HPGDALDH1A1MAOBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220143229-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-05-12 US disclosed
US-20220143229-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-05-12 US disclosed
US-11260136-B2 Radio-pharmaceutical complexes BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-03-01 US disclosed
US-20210322583-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER AS (NO) 2021-10-21 US disclosed
US-20210322583-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER AS (NO) 2021-10-21 US disclosed
CN-107278155-B Radiopharmaceutical complexes 拜耳有限公司 2021-03-30 CN disclosed
US-20190298865-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-03 US disclosed
US-20190298865-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-03 US disclosed
EP-3468619-A1 RADIO-PHARMACEUTICAL COMPLEXES Bayer Pharma Aktiengesellschaft (DE) 2019-04-17 EP disclosed
US-20190091354-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-03-28 US disclosed
WO-2017211809-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-12-14 WO disclosed
WO-2017211809-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-12-14 WO disclosed
US-20170340759-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER AS (NO) 2017-11-30 US disclosed
US-20170340759-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER AS (NO) 2017-11-30 US disclosed
US-20170340759-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER AS (NO) 2017-11-30 US disclosed
EP-3233137-A1 RADIO-PHARMACEUTICAL COMPLEXES Bayer AS (NO) 2017-10-25 EP disclosed
WO-2017162555-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-09-28 WO disclosed
WO-2017162555-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-09-28 WO disclosed
WO-2016096843-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER AS (NO) 2016-06-23 WO disclosed
WO-2016096843-A1 RADIO-PHARMACEUTICAL COMPLEXES BAYER AS (NO) 2016-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210322583-A1 RADIO-PHARMACEUTICAL COMPLEXES PTMS, THOP1, PHPT1 KDM4E 4009/4885HPGD 1440/4885ALDH1A1 3512/4885
US-20220143229-A1 RADIO-PHARMACEUTICAL COMPLEXES EGFR, MET, ERBB2 KDM4E 1959/4885HPGD 608/4885ALDH1A1 3506/4885
US-11260136-B2 Radio-pharmaceutical complexes EGFR, MET, ERBB2 KDM4E 2112/4885HPGD 531/4885ALDH1A1 3148/4885
US-20170340759-A1 RADIO-PHARMACEUTICAL COMPLEXES PTMS, THOP1, PHPT1 KDM4E 4022/4885HPGD 1420/4885ALDH1A1 3524/4885
US-20190091354-A1 RADIO-PHARMACEUTICAL COMPLEXES EGFR, MET, ERBB2 KDM4E 2143/4885HPGD 544/4885ALDH1A1 3158/4885
US-20190298865-A1 RADIO-PHARMACEUTICAL COMPLEXES FAP, PHPT1, DNPEP KDM4E 1459/4885HPGD 632/4885ALDH1A1 2075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.